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2-[(2,6-dichlorophenyl)methyl]-N-(furan-2-ylmethyl)-4-hydroxy-N-methylpyrimidine-5-carboxamide
N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(dimethyl-1,2-oxazol-4-yl)-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}acetamide
N-ethyl-2-{[(5-fluoropyridin-3-yl)carbamoyl]amino}propanamide
3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-(6-methoxypyrimidin-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4R)-1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(1,4-dioxan-2-ylmethyl)-N-methyl-1,3-oxazole-4-carboxamide
2,6-dimethyl-4-[2-(morpholin-4-ylmethyl)phenyl]phenyl acetate
N-[(3-chlorophenyl)methyl]-3-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]propanamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
2-{[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}morpholine
N-(2-methoxyethyl)-N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
2-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)ethan-1-ol
1-methyl-4-{5-[1-(2-phenylethyl)pyrrolidin-2-yl]thiophene-2-carbonyl}piperazin-2-one
2-chloro-4-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenol
N-phenyl-5-(1,3-thiazol-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(1R,5R)-6-[(2,5-dimethylphenyl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(cyclohex-1-en-1-ylmethyl)-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
6-ethyl-2-methoxy-3-{[(9H-purin-6-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
6-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
4-[(4-fluorophenyl)methyl]-1-(4-methyl-1,3-thiazole-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-butyl-N-methyl-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
4-(1H-imidazol-1-yl)-1-[3-(3-methylphenoxymethyl)piperidin-1-yl]butan-1-one
2-[3-fluoro-5-(2-methylpropoxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-(4-fluorophenyl)-5-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-1,3-thiazol-2-amine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-(2,4-dioxo-1,3-thiazolidin-3-yl)-N-methylacetamide
2-(3-methoxyphenyl)-1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{[4-(trifluoromethyl)phenyl]methyl}piperidine
N-(2-hydroxyethyl)-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-N-(thiophen-2-ylmethyl)benzamide
1-methyl-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
(4aS,8aS)-2-[(3,5-dichloropyridin-4-yl)methyl]-decahydroisoquinolin-4a-ol
2-{[4-(4-methoxy-3-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-methyl-1H-imidazole
2-ethyl-8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-butyl-N-(furan-2-ylmethyl)-3-(2-oxopiperidin-1-yl)propanamide
4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2,5-dimethylpyrimidine
8-[(2-aminopyridin-3-yl)methyl]-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-[2-(4-chlorophenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-1-methyl-N-(oxan-4-ylmethyl)-1H-indole-6-carboxamide
N-(1-carbamoylcyclopentyl)-2,3,6-trimethylquinoline-4-carboxamide
4-[2-(dimethylamino)-2-(3-fluorophenyl)acetamido]-N,N-dimethylbutanamide
(4S)-3-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-phenyl-1,3-oxazolidin-2-one
7-(1-benzothiophen-3-yl)-4-(2-methoxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(4-methoxyphenyl)methyl]-4-(quinoline-2-carbonyl)piperazin-2-one
N,N-dimethyl-6-{[1-(thiomorpholin-4-yl)hex-5-en-2-yl]oxy}pyrazin-2-amine
1-[(4aR,8aR)-7-[(2-fluoro-5-methoxyphenyl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
(4aS,8aR)-6-(5-methoxypyrimidin-2-yl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
methyl 4-{5-chloro-2-[(cyclopropylformamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]ethan-1-one
6-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}quinoxaline