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5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-{1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
1-cyclohexyl-4-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperazine
3-(aminomethyl)-4-(2,4-dimethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
ethyl 2-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-2-yl)acetate
2-fluoro-N-({3-methyl-7-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)benzamide
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-7-oxo-3-(5-oxopyrrolidine-3-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(furan-2-ylmethyl)-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
N-cyclopropyl-2,6-dihydroxy-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
N-(2-methoxyethyl)-1-{1-[3-(1H-pyrrol-1-yl)propanoyl]piperidin-4-yl}piperidine-3-carboxamide
N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-3-carboxamide
[1-(adamantan-1-yl)propan-2-yl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-{2-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
N-(2,1,3-benzothiadiazol-4-yl)-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine-1-carboxamide
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-2-(2-phenylethyl)piperidine
methyl 5-(cyclohexylamino)-3-acetamido-1-ethyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-2,3-dihydro-1-benzofuran-7-carboxamide
4-(1-butyl-1H-imidazol-2-yl)-1-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}piperidine
methyl 1-{2-hydroxy-3-[4-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
N-[(4-phenyloxan-4-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
N-(1-{7-[(2-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)propanamide
4-benzyl-3-ethyl-1-(1-ethyl-1H-pyrazole-3-carbonyl)-1,4-diazepan-5-one
(2S,4R)-1-(cyclopentylmethyl)-N,N-diethyl-4-(thiophene-2-amido)pyrrolidine-2-carboxamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
7-(1-benzothiophen-3-yl)-4-(furan-3-carbonyl)-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-5-methyl-2-phenyl-1H-imidazole-4-carboxamide
N-{1-[7-(4-tert-butylbenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-2-(dimethylamino)acetamide
2-(4-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}piperidin-1-yl)pyrimidine
3-methanesulfonamido-N-(3-phenylprop-2-yn-1-yl)-N-propylpropanamide
N-methyl-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-(1H-pyrazol-3-ylmethyl)acetamide
(1S,5R)-3-{2-[4-(dimethylamino)phenyl]acetyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
dimethyl[2-(2-{1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl}-1H-imidazol-1-yl)ethyl]amine
methyl 3-(2-methoxyacetamido)-5-[(pentan-3-yl)amino]-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-methoxy-3-({methyl[2-(2-oxopiperidin-1-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-(4-{[2-(propylamino)pyrimidin-5-yl]methyl}morpholin-3-yl)-N-(pyridin-3-yl)acetamide
4-cyclohexyl-3-{[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]methyl}-4H-1,2,4-triazole
1-methyl-4-{1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carbonyl}piperazin-2-one
1-(2-phenylethyl)-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2H-1,3-benzodioxol-5-ylmethyl)[(2-methoxypyrimidin-5-yl)methyl](pyridin-3-ylmethyl)amine
2-hydroxy-5-{[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}benzoic acid
6-(benzyloxy)-4-[(3-methylthiophen-2-yl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
N-(1-methyl-1H-1,2,3-triazol-4-yl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3-(2,5-dioxoimidazolidin-4-yl)propanamide
7-(1,3-benzothiazol-2-yl)-4-(pyrimidin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidin-2-amine
5-methyl-2-(4-{[5-(1H-1,2,4-triazol-5-ylsulfanyl)furan-2-yl]methyl}piperazin-1-yl)pyrimidin-4-amine
1-(2H-1,3-benzodioxol-5-yl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidin-4-amine
(3aR,6aS)-2-[(5-phenylthiophen-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole
2-(dimethylamino)-N-[2-(1H-imidazol-1-yl)ethyl]-2-(3-methylphenyl)acetamide
1-{1-[6-(cyclopentylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}propan-1-ol