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N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-methyl-1H-1,3-benzodiazole-7-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{4-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}methanol
3-ethyl-1-[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-3-ol
N-methyl-6-(morpholin-4-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrimidin-4-amine
3-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-N-(3-chloro-4-fluorophenyl)propanamide
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]propanamide
1-[1-(2-methylpropanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N,1-dimethyl-3-(2-methylpropyl)-N-[3-(pyrrolidin-1-yl)butyl]-1H-pyrazole-5-carboxamide
(1S,5R)-6-propyl-3-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{4-phenyl-1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-5-yl}benzonitrile
4-{[2-(ethylamino)pyrimidin-5-yl]formamido}-N,4-dimethylpentanamide
5-ethyl-4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-methylpyrimidine
(3S,4R)-3-methoxy-1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)piperidin-4-amine
5-[6-(dimethylamino)pyrimidin-4-yl]thiophene-2-carboxylic acid
(4aS,7aR)-1-(5-methylpyrazine-2-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclopentyl-4-(5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carbonyl)piperazine
N-(3-phenylpropyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N3-tert-butyl-4-oxo-N5-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-({1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-hydroxyazepan-4-yl}methyl)methanesulfonamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(quinoline-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-acetamido-N-(2-methoxyethyl)-3-methyl-N-[(4-methylphenyl)methyl]butanamide
3-ethyl-1-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}urea
4-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-1H-1,3-benzodiazole
(3R,4R)-4-(hydroxymethyl)-1-[3-(2-methylphenyl)benzoyl]piperidin-3-ol
2-(methylamino)-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)pyridine-4-carboxamide
3-benzyl-8-[(8-methoxyquinolin-2-yl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
4-(3-fluorophenyl)-N-methyl-N-[1-(pyridin-4-yl)ethyl]benzamide
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-(2-{7-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,4-dimethylbenzamide
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-propyl-1H-1,2,4-triazole
1-cyclohexyl-3-cyclopropyl-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
4-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-7-fluoro-1,2-dihydroquinolin-2-one
N-methyl-N-(2-phenylethyl)-2-[4-(propane-1-sulfonyl)morpholin-3-yl]acetamide
3-[2-(dimethylamino)ethyl]-5-{1-[3-(furan-2-yl)benzoyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
2-[(4-{4-[1-hydroxy-2-(morpholin-4-yl)ethyl]phenyl}-1H-pyrrolo[2,3-b]pyridin-6-yl)amino]ethan-1-ol
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-[3-(trifluoromethyl)phenyl]piperazine
N-[3-(1H-indazol-1-yl)propyl]-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
2-({2-[ethyl(3-methylphenyl)amino]ethyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-benzoyl-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazine
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(2-oxoazepan-1-yl)acetamide
N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-3-[(thiophen-2-ylmethyl)amino]benzamide
7-[(3-methoxyphenyl)methyl]-2-(2-methylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decane
N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-3-(3-methyl-1H-pyrazol-1-yl)-N-(pyridin-2-ylmethyl)propanamide
2-[(2-fluorophenyl)methyl]-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,3-benzoxazole-6-carboxamide
2-(1-methyl-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol