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ethyl 1-(1,3-benzothiazol-2-ylmethyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
N-[4-(1H-pyrazol-1-yl)phenyl]-1-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
N6-cyclobutyl-N5,N5-dimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-[4-(1H-pyrazol-5-yl)phenyl]-1-[(2,3,6-trifluorophenyl)methyl]piperidine-3-carboxamide
4-({2-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]amine
1-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
{4-[(4-chlorophenyl)methyl]-1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl}methanol
methyl(oxan-2-ylmethyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(2R,3R)-2-methoxy-1'-[(2-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
5-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}-2-(pyridin-2-yl)pyrimidine
N-cyclopropyl-2,3-dimethoxy-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]benzamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amine
2-ethyl-5-{[4-(2-phenylethyl)piperidin-1-yl]methyl}pyrimidine
1-(dimethyl-1,3-thiazole-4-carbonyl)-3-phenylpiperazine
(3S,4S)-1-(2,3-dihydro-1,4-benzodioxine-5-sulfonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
methyl 3-(2-methoxyacetamido)-1-methyl-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-acetamido-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)benzamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(3-methoxyphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
2-{4-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]piperidin-1-yl}acetamide
2-methoxy-6-(3-methoxy-6-methylpyridin-2-yl)-N,N-bis(propan-2-yl)benzamide
2-(1H-indol-3-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(5-methylfuran-2-yl)methyl]amine
(4-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-1-methylpiperazin-2-yl)methanol
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[2-(1H-pyrazol-1-yl)ethyl]amine
4-({2-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-({5-[(2-chloro-4-fluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
2-[(6-chloro-2H-chromen-3-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
N-methyl-3-(1-methylpiperidin-2-yl)-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}propanamide
(4aR,7aS)-1-ethyl-4-(pent-2-yn-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
N-[(2R,3R)-2-ethoxy-1'-[(4-oxo-4H-chromen-3-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
3-(4-fluorophenyl)-4-[5-(phenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-2-one
2-chloro-4-fluoro-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide
9-(3-methyl-1,2-oxazole-5-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(3,4,5-trimethoxyphenyl)ethan-1-one
1-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)piperidine-4-carboxamide
methyl 3-(2,2-dimethylpropanoyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2R)-2-amino-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-phenylacetamide
(4-{[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
1-(3-carbamoylpyridin-2-yl)-4-(2,3-dihydro-1H-inden-5-yloxy)piperidine-4-carboxylic acid
ethyl 1-(2-methoxyacetyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
1-{4-[(2-methylpropyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-[(4aR,7aS)-4-[(2-cyanophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
5-[1-(3-chlorothiophene-2-carbonyl)piperidin-4-yl]-3-[(2,3-dimethoxyphenyl)methyl]-5-methylimidazolidine-2,4-dione
7-(oxan-4-yl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
N-[1-(4-methoxyphenyl)-5-oxopyrrolidin-3-yl]-2-propyl-1,3-thiazole-4-carboxamide
3-{1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-2-yl}pyridine
N-[(3R,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide