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4-{[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]methyl}morpholine
(2-oxo-2-{6-[(thiophen-2-ylmethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}ethyl)urea
2-{3-[4-(4-methylphenoxy)piperidine-1-carbonyl]piperidin-1-yl}acetamide
1-[2-(4-fluorophenyl)ethyl]-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxylic acid
N-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-2-oxo-1,3-dioxa-8-azaspiro[4.5]decane-8-carboxamide
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(piperidin-4-yl)piperidine
2-(4-fluorophenyl)-2-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]ethan-1-ol
7-[(2,3-difluorophenyl)methyl]-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decane
4-(2-methyl-4-phenylpyrimidine-5-carbonyl)-2-(trifluoromethyl)morpholine
7-(6-fluoro-1H-1,3-benzodiazole-2-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[3-(dimethylamino)-1-phenylpropyl]-3-(2-fluoro-4-methoxyphenyl)urea
N-cyclopropyl-1-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
4-(2-fluoro-5-methylphenoxy)-1-(3-methylbut-2-enoyl)piperidine-4-carboxylic acid
N-[(3S,5S)-1-benzoyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
1-{4-[(4-{spiro[2.4]heptane-1-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperazin-1-yl}ethan-1-one
N-[2-(dimethylsulfamoyl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
1-(furan-2-ylmethyl)-N-{[2-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
4-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
methyl[(1-methyl-1H-pyrazol-4-yl)methyl][(4-{[1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
5-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
2-(2-{1-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
2-[5-({6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}methyl)furan-2-yl]benzonitrile
7-(3,6-dimethylpyrazin-2-yl)-4-(oxane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-hydroxy-1-(thian-4-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-(morpholin-3-yl)ethan-1-one
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2-chloro-5-({[(1-cyclopropyl-1H-imidazol-5-yl)methyl]carbamoyl}amino)-N-(propan-2-yl)benzamide
N-[2-(1H-imidazol-4-yl)ethyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-amino-5-{[1-phenyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydropyrimidin-4-one
1,3-dimethyl-5-({[4-methyl-4-(methylsulfanyl)pentan-2-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[3-(2-methoxyphenyl)propyl]-2-(1-methylpiperidin-2-yl)acetamide
6-methyl-14-[(1E)-1-phenylprop-1-en-2-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(3S,4S)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-{[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methyl}-1H-1,3-benzodiazole
8-[(2-aminopyridin-3-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methanesulfonamido-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]propanamide
3-(4-methoxyphenyl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-pyrazole-5-carboxamide
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-1-(2-methylpropyl)-1H-1,3-benzodiazole
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(4-phenylphenyl)propan-1-one
4-[2-(4-methoxyphenyl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-(4,5-dimethyl-1H-imidazol-1-yl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-methyl-N-(piperidin-3-ylmethyl)propanamide
N-(2-{7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
2-hydroxy-5-({[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amino}methyl)benzoic acid
1-[1-(4-amino-5-methylpyrimidin-2-yl)piperidin-4-yl]-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide