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(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
2-(4-chlorophenyl)-3-(pyrrolidine-1-carbonyl)pyridine
2-amino-4-[4-ethoxy-3-(hydroxymethyl)phenyl]-6-(6-methoxypyridin-3-yl)pyridine-3-carbonitrile
7-(2-cyclohexylethyl)-2-[5-(methoxymethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decane
4-{[5-chloro-3-methoxy-2-(propan-2-yloxy)phenyl]methyl}-1λ6-thiomorpholine-1,1-dione
5-(5-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)-1H-1,3-benzodiazole
5-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}pyridine-2-carbonitrile
ethyl 1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
N-[3-methyl-1-(pyridin-3-yl)butyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
(4aS,7aR)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl[(3-methylpyridin-4-yl)methyl]{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-(phenoxymethyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
3-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
4-chloro-2-fluoro-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
5-ethyl-1'-(4-methoxy-3-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-chloro-4-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}phenol
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(6-hydroxy-6-methylheptan-2-yl)-5-methoxybenzamide
N-(1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-4-yl)pyrimidin-2-amine
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperazin-1-yl)-1-(piperidin-1-yl)ethan-1-one
N-[(3S,4R)-4-(4-methoxyphenyl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrrolidin-3-yl]acetamide
N-(furan-2-ylmethyl)-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-(prop-2-en-1-yl)acetamide
(1S,4S)-2-(3,4-difluorophenyl)-5-[5-(4-methoxyphenyl)furan-2-carbonyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
1-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-(2-oxoazepan-3-yl)-2,3,4,9-tetrahydro-1H-carbazole-7-carboxamide
2-methoxy-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
ethyl 1-[(3-methoxyphenyl)methyl]-5-(1,2,5-thiadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{2-methyl-5-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]phenyl}imidazolidin-2-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]acetamide
(3aR,6aR)-2-[4-(4-fluorophenyl)-4-oxobutanoyl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl (2S,4S)-1-[(2-methylphenyl)methyl]-4-(pyridine-2-amido)pyrrolidine-2-carboxylate
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl][(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
1-benzyl-3-(2-methoxyethyl)-8-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-{1-[3-(1H-pyrazol-4-yl)benzoyl]piperidin-4-yl}pyrimidin-4-ol
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-amine
1-(4-fluorophenyl)-3-[3-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrrolidine
2-methoxy-1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
dimethyl({[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl](3-methylphenyl)methyl})amine
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N-methyl-N-(propan-2-yl)acetamide
3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1-(5,7,8-trimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
N-{1-[7-(3-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclopropanecarboxamide
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
4-({1-[2-(1H-imidazol-5-yl)ethyl]-5-(5-methylthiophen-2-yl)-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
2-[4-(4-methyl-1H-pyrrole-2-carbonyl)piperazin-1-yl]-1,3-benzothiazole
N,1-dimethyl-3-(thiomorpholine-4-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N3-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-N5-[2-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide