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3-{2-[4-(3-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
5-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
6-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-(4-methoxybenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-amine
5-chloro-N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
3-(1-acetylpiperidin-3-yl)-1-(4-benzylpiperazin-1-yl)propan-1-one
4-[4-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]aniline
2-(3-methoxyphenyl)-1-{5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}azetidine
4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[2-(2-ethoxyethoxy)phenyl]-3-{1-oxaspiro[4.4]nonan-3-yl}urea
1-{[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
3-(azepane-1-carbonyl)-N-[(4-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{4-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
(2S)-N-[3-(1H-pyrazol-1-yl)phenyl]-1-[3-(pyridin-3-yl)propyl]pyrrolidine-2-carboxamide
(1S,5R)-6-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-N-(propan-2-yl)pyrimidin-4-amine
methyl 3-{[4-(furan-2-carbonyl)-7-oxo-1,4-diazepan-1-yl]methyl}benzoate
(benzylsulfamoyl)[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amine
(4aS,8aR)-6-(1-aminocyclobutanecarbonyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(2H-1,3-benzodioxol-5-yl)-N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
(1R,5R)-6-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(3aS,6aR)-5-[(6-methylpyridin-2-yl)methyl]-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(3-hydroxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(5-chlorothiophene-2-carbonyl)-4-(2,6-dimethylpyridin-4-yl)piperazine
methyl 3-(2-chloro-6-fluorobenzamido)-6-{[(2-methoxyethyl)(propan-2-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
2-(4-fluorophenoxymethyl)-N-[2-(pyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
N,5-dimethyl-4-[(pyridin-2-ylmethyl)amino]-N-(thiophen-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(furan-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[2-({1-[(6-chloroquinolin-2-yl)methyl]piperidin-4-yl}oxy)ethyl]dimethylamine
3-[4-phenyl-5-(quinolin-4-yl)-1H-imidazol-1-yl]propan-1-ol
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylpiperidine-4-carboxamide
4-(4-fluorophenyl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-4-oxobutanamide
N-methyl-2-[4-(4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-ylmethyl}-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyrimidin-4-amine
4-benzyl-1-(2-{1-methyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-oxoethyl)pyrrolidin-2-one
1-(1-pentanoylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
ethyl 2-(1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
1-(3-chloro-4-methoxyphenyl)-3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]urea
2-{4-[1-(3-fluoropropyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}pyridine
1-{2-[({4-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)amino]ethyl}imidazolidin-2-one
2-chloro-N-{2-[(1-phenyl-1H-1,2,3-triazol-4-yl)formamido]ethyl}benzamide
N-[4-(azepan-1-yl)butyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-[1-(furan-3-ylmethyl)piperidin-4-yl]propanamide
1-(4-{2-[7-(3-chlorophenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
7-{4-[1-(piperidin-1-yl)ethyl]phenyl}-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine