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1-{4-[4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]phenyl}ethan-1-one
(1S,5R)-3-[2-(2-methylphenyl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-cyclohexylpiperazin-2-one
2-amino-2-methyl-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
N-methyl-3-(5-methylthiophen-2-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-pyrazole-5-carboxamide
4-(naphthalen-2-yloxy)-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
N-(1-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
2-{9-[(2,3-dimethoxyphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
2-(furan-2-yl)-5-(1-{[1-(propan-2-yl)piperidin-4-yl]methyl}-1H-imidazol-2-yl)pyrimidine
4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]-1-[1-(methylsulfanyl)propan-2-yl]piperidine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
methyl 4-({4-[1-(4-chlorophenyl)cyclopropanecarbonyl]-7-oxo-1,4-diazepan-1-yl}methyl)benzoate
6-[4-(1H-imidazol-1-yl)benzoyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-6-azaspiro[2.5]octane-1-carboxamide
4-cyclohexyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)-1,4-diazepane-1-carboxamide
2-(3-chloro-4-hydroxyphenyl)-N-[2-(2-ethoxyphenoxy)ethyl]-N-methylacetamide
N-methyl-N-(1,2-oxazol-5-ylmethyl)-2-(3-phenylpiperidin-1-yl)acetamide
N-{1-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]propan-1-ol
4-benzyl-3-butyl-1-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1-methoxypropan-2-yl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-methyl-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}quinoxaline
N4-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrimidine-2,4-diamine
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
1-(2,3-dihydro-1H-inden-2-yl)-4-[5-(methoxymethyl)furan-2-carbonyl]-1,4-diazepane
1-methyl-1-(1-methylpyrrolidin-3-yl)-3-(2-phenyl-1,3-benzoxazol-5-yl)urea
(3R,4R)-4-(azepan-1-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-ol
3-(7-methyl-1H-indol-3-yl)-4H-chromen-4-one
N-[(2-fluorophenyl)methyl]-2-[(1-methylpiperidin-4-yl)(pyridin-3-ylmethyl)amino]acetamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
8-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-1-(pyrrolidin-1-yl)cyclohexane-1-carboxamide
methyl[2-methyl-3-(pyrrolidin-1-yl)propyl][(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
6-methyl-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-2-phenylpyrimidin-4-amine
N-(2-{4-[(1-ethyl-1H-indol-5-yl)methyl]morpholin-2-yl}ethyl)acetamide
2-{[(furan-2-ylmethyl)(prop-2-en-1-yl)amino]methyl}benzoic acid
4-(4-chlorophenyl)-1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}butan-1-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
3-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)pyridin-2-amine
{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,5-dihydro-1H-pyrrol-2-yl}methanol
N-(2,3-dihydroxypropyl)-4-ethyl-N,2-dimethyl-1,3-thiazole-5-carboxamide
9-(1-aminocyclopropanecarbonyl)-2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
3-cyclohexyl-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1H-pyrazole-4-carboxamide
4-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)benzoyl]thiomorpholine
N-butyl-2-(4-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
[4-({1-[2-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
(3S,4S)-4-cyclopropyl-1-[(2-methylpyrimidin-5-yl)methyl]pyrrolidine-3-carboxylic acid
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-(1,3-thiazol-2-yl)piperazine
1-(2,3-dihydro-1H-inden-2-yl)-4-[(2-methyl-5-propylpyrimidin-4-yl)amino]pyrrolidin-2-one