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N-[4-(4-{[2-(1H-indol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-2-phenoxyacetamide
1-{4-[({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]phenyl}pyrrolidin-2-one
1-(2-methoxyethyl)-3-(2-methylpropyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-methyl-1-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]-1,4-diazepan-5-one
3-methoxy-1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
2-ethyl-6-(2-methoxy-4-methylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-{[3-(methylsulfanyl)phenyl]methyl}-N-(propan-2-yl)morpholine-2-carboxamide
5-cyclopropanecarbonyl-1'-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(2-methoxyethyl)-4-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
{1-[(3-methylthiophen-2-yl)sulfonyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-5-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
5-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
6-amino-N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)pyridine-3-carboxamide
6-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidine-1-carbonyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)azetidin-3-yl]-2-methylpiperidine
4-chloro-2-({3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}methyl)phenol
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(1H-pyrazole-3-carbonyl)piperidine
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyrrolidine-1-carbonyl)piperidine
1-{2-oxo-2-[3-(4-phenylbenzoyl)piperidin-1-yl]ethyl}pyrrolidin-2-one
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
2-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-5-methylpyrazine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
ethyl 2-{[2-(trifluoromethyl)morpholine-4-carbonyl]amino}benzoate
{1-[3-(naphthalen-1-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-4-yl}(thiophen-2-yl)methanol
N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
6-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
1-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-3-methyl-3-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]urea
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl]methanol
N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyrrolidin-1-yl)acetamide
1-[(4-methoxyphenyl)methyl]-4-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
5-(3-fluorophenoxymethyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
4-(4-ethoxy-3-methylphenyl)-N-[3-(pyridin-3-yl)propyl]butanamide
N-(2-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
4-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1,3-oxazole-5-carboxamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-{[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-ethyl-1,2,4-oxadiazole
1-cyclopentyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-6-oxopiperidine-3-carboxamide
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-ethyl-N-methylacetamide
(1R,3S)-3-{[2-(4-phenylpiperidin-1-yl)ethyl]carbamoyl}cyclopentane-1-carboxylic acid
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[2-methoxy-1-(pyridin-2-yl)ethyl]acetamide
1-[(2,3-difluorophenyl)methyl]-3-{[(1,3-dihydroxypropan-2-yl)amino]methyl}-3-hydroxypiperidin-2-one
1-methyl-4-({4-methyl-5-[1-(pyridine-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
2-(2-hydroxypropyl)-9-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-4-{3-methyl-5-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazol-1-yl}piperidine
2-({4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}methyl)benzoic acid
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]propan-1-one
2-ethoxy-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(quinoline-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one