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ethyl 1-(4-methylphenyl)-5-({[2-(1H-1,2,4-triazol-1-yl)ethyl]amino}methyl)-1H-pyrazole-4-carboxylate
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-(prop-2-en-1-yl)-4-[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperazine
(1S,5R)-6-(1-methyl-1H-indole-3-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-4-methylpiperidine-4-carboxamide
N-[2-(3-methoxyphenyl)ethyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-[4-(1H-pyrazol-1-yl)phenyl]-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxamide
N-benzyl-N,1-dimethyl-5-({[4-(trifluoromethoxy)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[2-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
N-(1,3-benzothiazol-2-ylmethyl)-2-(dimethylamino)-6-(2-methylphenyl)pyridine-3-carboxamide
(1H-indol-5-ylmethyl)(methyl)(pyrazin-2-ylmethyl)amine
1-(4-benzylpiperazine-1-carbonyl)-6-[(2,4-difluorophenyl)methyl]-6-azaspiro[2.5]octane
(1S,5R)-1,3,3-trimethyl-6-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}-6-azabicyclo[3.2.1]octane
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
N-(furan-2-ylmethyl)-3-{spiro[indene-1,4'-piperidine]-1'-yl}propanamide
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2-(ethylamino)pyrimidine-5-carboxamide
(3S,4R)-4-(pyridin-4-yl)-1-(4,4,4-trifluorobutanoyl)pyrrolidine-3-carboxylic acid
2-(2-methoxyphenyl)-4-[(3-methylquinoxalin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(1H-pyrazol-1-yl)benzamide
6-[(3,4-dimethoxyphenyl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(propan-2-yloxy)ethan-1-one
2-methyl-N-(1-{7-[(6-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
1-cyclopentyl-3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-butyl-8-[4-(morpholin-4-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[(3S,4S)-1-(4-ethenylbenzoyl)-3-hydroxypiperidin-4-yl]methyl}-3-methylbutanamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-(methylsulfanyl)acetamide
8-[(2-fluorophenyl)methyl]-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(pyridin-3-ylmethyl)-N-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
1-{4-[(4-chloro-3-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
4-[(3-methoxyphenyl)methyl]-1-[1-(2-phenylethyl)piperidin-4-yl]-1,4-diazepan-5-one
1-(furan-2-ylmethyl)-3-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]urea
2-methoxy-1-(4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N,N-dimethyl-5-{[5-oxo-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}furan-2-carboxamide
4-(1-{4-[3-(4H-1,2,4-triazol-4-yl)phenyl]phenyl}ethyl)morpholine
N-(2-{3-methyl-7-oxo-7H-[1,3]thiazolo[3,2-b][1,2,4]triazin-6-yl}phenyl)-6-oxo-1,6-dihydropyridine-2-carboxamide
(3aR,6aR)-2-(cyclohexylcarbamoyl)-5-(3-methoxypropyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2H-1,3-benzodioxol-5-yl)-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
3-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-benzyl-1-[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
ethyl 4-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine-1-carboxylate
2-amino-4-methyl-N-[(2-methylphenyl)(pyridin-4-yl)methyl]pyrimidine-5-carboxamide
4-(piperidin-1-yl)-1-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazin-1-yl}butan-1-one
4-(1,3-benzothiazol-2-yl)-2-({[2-(3,4-dimethoxyphenyl)ethyl]amino}methyl)phenol
[(1R,3S,3aS,6aR)-3-(4-chlorophenyl)-1-ethyl-5-methyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
2-(adamantan-1-yl)-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}acetamide
3-(2-chlorophenyl)-3-{2-[4-(2,4-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-1-methylpyrrolidine-2,5-dione
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-4-carboxamide