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1-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidin-3-ol
N-[2-(dimethylsulfamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-1-phenylcyclopropane-1-carboxamide
3-[1-(2,7,8-trimethylquinoline-4-carbonyl)pyrrolidin-2-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{3-oxo-3-[3-oxo-4-(2-phenylphenyl)piperazin-1-yl]propyl}acetamide
4-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[(7-fluoroquinazolin-4-yl)amino]-1-(2-methoxyphenyl)pyrrolidin-2-one
N-ethyl-3-(4-methoxyphenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
methyl 2-({4-[1-(2-acetamidoacetyl)piperidin-3-yl]-5-(4-fluorophenyl)pyrimidin-2-yl}sulfanyl)acetate
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}pyrrolidine-2,5-dione
N,2-dimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-(1H-imidazol-2-ylmethyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
(3aS,6aS)-2-[(2-chlorophenyl)methyl]-5-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
13-[4-(diethylamino)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
2-butyl-8-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N,N,4-trimethyl-3-({[2-(propan-2-yloxy)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(3S,4S)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]-4-(propan-2-yloxy)pyrrolidin-3-ol
N-[4-(1H-pyrazol-1-yl)phenyl]-2-[2-(pyridin-2-yl)ethyl]piperidine-1-carboxamide
(2S,4R)-N-(2-methoxyethyl)-4-{[(3-phenoxyphenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
ethyl 2,4-dimethyl-5-(3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidine-1-carbonyl)-1H-pyrrole-3-carboxylate
(2S)-1-[5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-methyl-2-phenylpiperazine
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
1-ethyl-4-({methyl[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}methyl)pyrrolidin-2-one
2-methyl-9-[(4-methyl-1,3-thiazol-5-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
N-cyclooctyl-2-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]acetamide
3-[3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carbonyl]-2H-chromen-2-one
(1-{1-[4-(4-methylphenyl)phenyl]piperidin-4-yl}pyrrolidin-3-yl)methanamine
1-[3-(dimethylsulfamoyl)-5-{[(4-methyl-1H-imidazol-5-yl)methyl]amino}benzoyl]piperidine-3-carboxamide
2-(2-methoxy-4-{12-oxo-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-14-yl}phenoxy)acetamide
1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
2-(1,2-oxazole-5-carbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(furan-2-yl)-2-hydroxyethyl]-3-(trimethyl-1H-pyrazol-4-yl)urea
5-fluoro-1,3-dimethyl-2-(3-methyl-1H-1,2,4-triazol-5-yl)-1H-indole
8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(4-chlorophenyl)-8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
N-{3-[4-({2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}amino)piperidin-1-yl]phenyl}pyridine-3-carboxamide
N-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
2-(3,4-dimethoxyphenyl)-1-{7-[hydroxy(pyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
N-butyl-6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-[4-(2-cyanophenyl)-3-oxopiperazine-1-carbonyl]piperidine-1-carboxamide
ethyl (2S)-2-[5-(2,6-dimethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propanoate
N-[2-(2,4-dimethoxyphenyl)ethyl]-1-(diphenylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(6-methylpyridin-2-yl)methyl]-2-(methylsulfanyl)pyrimidin-4-amine
4-(2-hydroxy-2-phenylacetyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
N-methyl-1-(naphthalen-1-ylmethyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
5-acetyl-N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]pyrimidin-2-amine
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-methylacetamide
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(quinolin-6-ylmethyl)amine