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N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(methylsulfanyl)acetamide
(4aR,7aS)-1-benzyl-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[2-(2-aminoethyl)quinazolin-4-yl](butyl)amino}butan-1-ol
5-tert-butyl-1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
5-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-4-methyl-1,3-oxazole
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
2-[9-(3-chlorobenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
2-methoxy-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
3-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl)amino]methyl}-5-methyl-1H-indole-2-carboxylic acid
1-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2H-1,3-benzodioxol-5-yl)-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)acetamide
2-[(3-methoxyphenyl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}morpholine
1-ethyl-N,3-dimethyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
methyl 3-(2-methoxybenzoyl)-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
7-(methylsulfanyl)-3-[(3-oxo-1,4-diazepan-1-yl)methyl]-1,2-dihydroquinolin-2-one
2-[benzyl(methyl)amino]-N-(pyridin-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)-N-methylacetamide
N-benzyl-N-(cyclopropylmethyl)-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
(5-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol
3-phenyl-N-{3-[2-(pyridin-2-yl)acetamido]phenyl}propanamide
5-methyl-N-[(1-methylpiperidin-4-yl)methyl]-1-[4-(pyridin-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-methoxyethan-1-one
2-[ethyl({[(3R,4R)-1-(2-ethylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[4-({3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-methoxyphenoxy)piperidine
N-({7-[3-(3-methoxyphenyl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
N-{2-[(1R,7S)-4-oxo-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-3-yl]ethyl}acetamide
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-[(2E)-3-phenylprop-2-en-1-yl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(4-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
1-[4-(benzyloxy)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N,2,3-trimethyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]quinoxaline-6-carboxamide
2-{4-[(6-methylpyridin-2-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N-methyl-3-(1H-1,2,3,4-tetrazol-1-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
2-methyl-5-(3-{[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
1'-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(4-methoxyphenyl)-4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-2-one
4-ethyl-1-(1H-indole-2-carbonyl)-1,4-diazepan-5-one
4'-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-(6-methoxy-2H-1,3-benzodioxol-5-yl)urea
1'-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]
N-benzyl-N-methyl-2-({[(2-methyl-1,3-thiazol-5-yl)methyl]amino}methyl)-2,3-dihydro-1H-inden-2-amine
methyl 4-(5-methyl-4-{[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}-1,3-oxazol-2-yl)benzoate
N,N-diethyl-3-methyl-4-{[methyl(oxan-2-ylmethyl)carbamoyl]amino}benzamide
8-methoxy-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
8-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N'-(adamantan-1-yl)-N-[2-(1H-imidazol-4-yl)ethyl]propanediamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(piperidin-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
3-(2,5-dioxoimidazolidin-4-yl)-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]propanamide