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1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
4-{[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-N-methylbenzamide
1-cyclopropanecarbonyl-N-[1-(pyrazin-2-yl)propan-2-yl]piperidine-4-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(2,3-dihydro-1H-inden-1-yl)acetamide
(4aR,7aS)-1-acetyl-4-(3-methyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-1-(1H-indole-6-carbonyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyridin-2-amine
N-{[7-(naphthalen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine-2-carboxamide
[(2-chlorophenyl)methyl]({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
8-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(2,3-dimethyl-1H-indole-5-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1-methyl-1H-imidazol-2-yl)(1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)methanol
3-(2-{[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}propyl)-3,4-dihydroquinazolin-4-one
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
dimethyl(2-{2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(3-fluorophenyl)methyl]piperidine
methyl 5-[(butan-2-yl)amino]-3-(furan-2-amido)-1-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(propan-2-yl)-1-[(1s,4s)-4-{[(2,5-dimethoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
methyl 5-(2,3-dihydro-1H-inden-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-(furan-3-yl)-2-(4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[2-(ethylsulfanyl)ethyl]pyrimidin-2-amine
methyl 6-[2-(4-fluorophenyl)acetyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methylacetamide
2-amino-4-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-(propan-2-yl)pyridine-3-carbonitrile
3-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-2-yl)pyridine
3-methyl-3-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1-[3-(pyridin-3-yl)phenyl]urea
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(propan-2-yloxy)ethyl]propanamide
3-({1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
3-{[1-(cyclohex-1-en-1-yl)ethyl]carbamoyl}-5-methoxybenzoic acid
1-(4-methylphenyl)-4-[2-(methylsulfanyl)pyridine-3-carbonyl]piperazin-2-one
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-(4-chloro-2-methylphenoxy)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}propanamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methyl-1H-pyrrole-3-carboxamide
4-phenyl-N-(1-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
N-(1-hydroxybutan-2-yl)-2-(4-hydroxyphenyl)-N-(thiophen-2-ylmethyl)acetamide
1-(2-chlorobenzoyl)-3-(2-methoxyphenoxy)azetidine
2-butyl-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1,3-benzoxazole-5-carboxamide
3-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-5-carboxamide
N-methyl-5-({4-[1-(4-methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
2-(1-ethylpiperidin-4-yl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(thiophen-2-yl)ethyl]propanamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(1,2-oxazol-3-ylmethyl)propanamide
N-[4-(3-fluorophenyl)phenyl]-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidine-3-carboxamide
N-[2-(1H-indol-3-yl)ethyl]oxane-2-carboxamide
methyl 5-(cyclopentylamino)-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2,4-difluorophenyl)-3-[(3-hydroxyazetidin-1-yl)sulfonyl]benzamide