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3-{[1-(3-aminobenzoyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(6-methyl-2H-1,3-benzodioxol-5-yl)-4-(1H-pyrrole-2-carbonyl)piperazine-1-carboxamide
[(3R,5R)-1-(7-methyl-1-benzofuran-2-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-{5-[2-(methoxymethyl)pyrimidin-5-yl]-4-phenyl-1H-imidazol-1-yl}acetic acid
1-methyl-2-oxo-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
(2S,4S)-4-amino-N-ethyl-1-[3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanoyl]pyrrolidine-2-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[3-(pyridin-3-yl)propanoyl]piperidine-4-carboxylic acid
2-methoxy-N-({5-[(2,3,5-trifluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
3-[({[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)methyl]piperidin-3-ol
1-(4-benzylpiperazine-1-carbonyl)-6-[(2,6-difluorophenyl)methyl]-6-azaspiro[2.5]octane
1-methanesulfonyl-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
3-(3-fluorophenyl)-N-[1-(1H-indol-2-yl)ethyl]-N-methyl-1H-pyrazole-4-carboxamide
2-methyl-3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indol-4-one
9-(3-methyl-1H-pyrazole-5-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3-methylphenyl)methyl]-2-(2-oxoazepan-1-yl)-N-(oxolan-2-ylmethyl)acetamide
1-[1-(2-methyl-1H-1,3-benzodiazole-6-carbonyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
N-{1-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2-(1H-1,2,4-triazol-3-yl)benzamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
3-chloro-5-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-(3-methoxypropyl)-3-(2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)-3-(2-methylphenyl)pyrrolidine-2,5-dione
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-[(1-propyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](prop-2-en-1-yl)(prop-2-yn-1-yl)amine
(3aS,6aS)-2-(carboxymethyl)-5-[(4-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
4-(2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)piperazin-2-one
1-cyclopentyl-5-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}piperidin-2-one
3-(3,6-dimethylpyrazin-2-yl)-4H-chromen-4-one
9-[2-(4-methylphenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1'-(2,3-dihydro-1H-inden-2-yl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-benzyl-8-[(3-chloro-4-hydroxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(3S)-3-ethyl-4-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]morpholine
[(3R,4R)-1-(1H-indole-6-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]pyridine
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(1H-1,2,4-triazol-1-yl)benzamide
1-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-6-ol
4-methoxy-6-[4-(3-methylpyridin-4-yl)piperazin-1-yl]pyrimidine
1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine
2,3-dimethyl-5-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1H-indole
N,1-dimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-5-(thiophen-2-yl)-1H-pyrazole-3-carboxamide
methyl 2-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole-4-carboxylate
2-(2H-1,2,3-benzotriazol-2-yl)-1-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]ethan-1-one
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1-(5-methanesulfonyl-2-methylphenyl)-3-methylurea
4-[(3-methylbut-2-en-1-yl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
1-benzyl-5-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3R,4R)-1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-6-(methoxymethyl)pyrimidin-4-amine
4-[1-(1H-imidazole-5-carbonyl)piperidin-4-yl]thiomorpholine
N-{2-[4-({[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}thiophene-3-carboxamide