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1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N-({7-[2-(3-fluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
N-[5-(3-chloro-4-methoxyphenyl)pyridin-2-yl]acetamide
5-(4-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)-6-phenyl-2,3-dihydropyridazin-3-one
1'-[(3-methylquinoxalin-2-yl)methyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(1R,5R)-6-benzyl-3-(3-phenyl-1,2-oxazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
[4-({[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl](methyl)amino}methyl)oxan-4-yl]methanol
methyl[(3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,2-oxazol-5-yl)methyl](2-phenylethyl)amine
2-methyl-4-[4-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)phenyl]butan-2-ol
4-[1-(2-phenylethyl)piperidin-4-yl]pyridine
3-[(3S,4R)-1-benzyl-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[2-(4-methoxyphenyl)ethyl]propanamide
methyl 4-{[4-fluoro-3-(2-methylpropanamido)phenyl]carbamoyl}piperazine-1-carboxylate
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-N-[2-(diethylamino)ethyl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-2,1,3-benzoxadiazole
2-phenoxy-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl](methyl){2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
1-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)-4-methylpiperazine
(1S,5R)-6-[4-(2-methylpropyl)benzoyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}acetamide
3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-2,6-dimethylquinoline
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
4-methyl-6-(3,4,5-trimethoxyphenyl)-1,2-dihydroquinolin-2-one
2-{4-[(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenoxy}ethan-1-ol
N-(1H-indol-2-ylmethyl)-2-[(3-methoxyphenyl)amino]butanamide
6-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-2-carbonitrile
1-(2-{[ethyl(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)-2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
1-[4-({ethyl[(1-methylpyrrolidin-3-yl)methyl]amino}methyl)phenyl]ethan-1-one
3-[3-(4-methylphenyl)-3-phenylpropanamido]propanoic acid
N-[(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane
N-(1-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
2-[4-(hydroxymethyl)phenyl]-2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]acetic acid
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-[3-(trifluoromethyl)phenyl]acetamide
5-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3,5-dimethyl-4,5-dihydro-1,2-oxazole
N-{2-[(4-fluorophenyl)carbamoyl]ethyl}-2-methyl-2-(thiophen-2-ylformamido)propanamide
4-({4-methyl-5-[1-(2-phenoxyethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
(2S,4S)-N-ethyl-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-1-phenylpiperidin-4-amine
1-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indazole
5-{2-[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
[(2S)-1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
(3S,9aR)-3,8-dibenzyl-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-amine
5-acetyl-2,4-dimethyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1H-pyrrole-3-carboxamide
1-[4-({[(2-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
3-[2-(dimethylamino)ethyl]-5-[1-(2-phenoxyacetyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione