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1-(benzyloxy)-8-[2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
N-{4-[2-(4,5-dimethylfuran-2-yl)-1H-imidazol-1-yl]-2-methoxyphenyl}acetamide
[(2,3-difluorophenyl)methyl](methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
1-(4-hydroxyphenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-5-oxopyrrolidine-3-carboxamide
5-[4-(cyclobutylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-N-methylpyrimidin-2-amine
1-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
2-(2,4-dimethylbenzenesulfonamido)-N-methyl-N-[2-(pyrrolidin-1-ylmethyl)propyl]acetamide
2-cyclopropyl-6-methyl-3-[4-(4-methylphenyl)piperazine-1-carbonyl]-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-methyl-4-(2-methyl-1H-imidazol-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}butanamide
1,9-dimethyl-4-(2-methyl-5-propylpyrimidin-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-(4-methylphenyl)propanamide
1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
N,6-dimethyl-2-propyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine
N-benzyl-3-[2-(methylsulfanyl)benzoyl]piperidine-1-carboxamide
N-{3-[(2-ethylphenyl)carbamoyl]phenyl}-2,5-dihydro-1H-pyrrole-2-carboxamide
{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
2-{4-[5-(2-methyloxan-2-yl)-1,2,4-oxadiazol-3-yl]phenyl}ethan-1-ol
2-({1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-4-methyl-1H-imidazole
2-{2-[6-amino-5-cyano-4-(4-methyl-1H-imidazol-5-yl)pyridin-2-yl]phenoxy}acetamide
2-(4-fluorophenoxy)-1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
(1H-1,3-benzodiazol-2-ylmethyl)[(2,3,5-trimethyl-1H-indol-7-yl)methyl]amine
methyl 5-(cyclohexylamino)-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-amino-7-[2-(dimethylamino)-2-(4-methylphenyl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[2-(3,4-dimethoxyphenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
3-{1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
1-ethyl-4-{[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-1H-pyrrole-2-carbonitrile
4-methyl-2-{1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
3-methoxy-N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N'-cyclopentyl-N-(propan-2-yl)butanediamide
2-{1-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]azetidin-3-yl}pyridine
methyl 9-(oxan-2-ylmethoxy)-7-oxo-3-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[5-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
(2R,3R,6R)-3-phenyl-5-(pyrrolidine-1-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-cyclopentyl-3-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
2-[3-(2-methoxyphenoxy)azetidin-1-yl]pyrazine
(3aR,6aR)-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-[1-(1,4-dioxan-2-ylmethyl)-1H-imidazol-2-yl]-1-methyl-1H-imidazole
2-[2-(4-chlorophenoxymethyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
3-(4-methylpiperazin-1-yl)-N-(4-phenoxyphenyl)pyrrolidine-1-carboxamide
N-(4-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}phenyl)acetamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzothiazole
N-[1-(7-{[5-(3-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-methoxypropanamide
5-(3-fluorophenoxymethyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazole-3-carboxamide
5-[1-(4-chlorophenyl)cyclobutanecarbonyl]-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(4-fluoro-2-methylphenyl)-3-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}propanamide
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxybutan-1-one