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1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-2-(methylsulfanyl)ethan-1-one
(1R,5S,6S)-N-(2-hydroxyethyl)-N-methyl-3-{[4-(methylsulfamoyl)phenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
4-acetamido-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(pyridin-3-yl)propan-2-yl]propanamide
ethyl 1-[(2-methoxyphenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
N-methyl-3-(1H-1,2,3,4-tetrazol-1-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]propanamide
2-[9-acetyl-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]pyridine-3-carbonitrile
N-[furan-2-yl(phenyl)methyl]-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-{[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzenesulfonamide
4-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]-5-ethylpyrimidin-2-amine
methyl({1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-2-phenylethyl})(pyridin-4-ylmethyl)amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-4-(1H-1,2,4-triazol-3-yl)benzamide
2-amino-6-cyclobutyl-4-[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
2-(4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}morpholin-3-yl)-1-(thiomorpholin-4-yl)ethan-1-one
1-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]-2-(dimethylamino)-2-(3-methylphenyl)ethan-1-one
1-{[5-(methoxymethyl)furan-2-yl]methyl}-3-[4-(methylsulfanyl)benzoyl]piperidine
8-chloro-2-({[(2-ethyl-1,3-thiazol-4-yl)methyl]amino}methyl)quinolin-4-ol
5-[1-(3,4-dimethylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-3,4-dihydropyrimidin-4-one
(1S,4S)-2-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2-azabicyclo[2.2.1]heptane
N-cyclopropyl-2-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}acetamide
6-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyridine-2-carbonitrile
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
1-{1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-4-phenylbutane-1,4-dione
{2-[(3S,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-1-yl]-1,3-thiazol-4-yl}methanol
N-cyclopentyl-3-{[(5-methyl-1H-pyrazol-3-yl)methyl]sulfamoyl}benzamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
7-methoxy-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-cyclopropyl-3-[(3-phenylpiperazin-1-yl)sulfonyl]benzamide
1-[(2-cyclohexylpyrimidin-5-yl)methyl]-3-ethylpiperidine-3-carboxamide
1-ethyl-N-[2-(2-fluorophenyl)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}thiomorpholine
N5-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-8-methylimidazo[1,2-a]pyridine-2-carboxamide
N-(1-methyl-1H-1,2,3-triazol-4-yl)-2-phenylazetidine-1-carboxamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
5-(1-ethyl-1H-pyrazol-3-yl)-1-(2-fluorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazole
(2S,4S)-N-ethyl-1-(1H-imidazol-4-ylmethyl)-4-[2-oxo-2-(piperidin-1-yl)acetamido]pyrrolidine-2-carboxamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3,3,3-trifluoropropan-1-one
2-(1-{1-phenylspiro[2.4]heptane-1-carbonyl}azetidin-3-yl)pyridine
3-[2-(2-fluorophenyl)ethyl]-1-(1,3-thiazol-2-yl)piperidine
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
N-(3-fluorophenyl)-3-[methyl(quinolin-3-ylmethyl)amino]propanamide
1-(1-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
methyl 2-{2-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}acetate
3-(4-tert-butylbenzoyl)-1-(1,2-oxazol-3-ylmethyl)piperidine
3-(1H-imidazol-2-ylmethyl)-6,7-dimethoxy-3,4-dihydroquinazolin-4-one