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N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methyl-1,3-thiazole-4-carboxamide
N-{1-[(4-fluorophenyl)methyl]-7-[2-(methoxymethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
1-[2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
4-[3-(5-benzyl-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
N-methyl-5-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(thiophen-2-ylmethyl)acetamide
7-{2-[(4-methylphenyl)methyl]benzoyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
5-methyl-1-propyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
4-{5-[2-(1H-imidazol-2-yl)benzoyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
N-cyclopropyl-1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
2-(furan-2-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(azepan-1-yl)-3-(3-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
2-[2-(dimethylamino)ethyl]-8-[2-(2-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(5-methyl-1H-indol-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}benzonitrile
N-benzyl-N-(cyclopropylmethyl)-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
7-(cyclohexylmethyl)-2-(5-methyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(5-acetylthiophen-3-yl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylacetamide
5-(2,4-difluorophenoxymethyl)-N-[3-(pyridin-3-yl)propyl]-1,2-oxazole-3-carboxamide
2-(4-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)phenol
1-[3-(4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine-1-carbonyl)phenyl]imidazolidin-2-one
2-[4-(cyclopropylmethyl)-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2,3-dihydro-1-benzofuran-5-carboxamide
(1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)methanol
2-[4-(2-amino-6-methoxypyrimidin-4-yl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
2-benzyl-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-1,3-thiazole-4-carboxamide
5-(2,4-difluorophenoxymethyl)-N-[2-(2-fluorophenyl)ethyl]-1,2-oxazole-3-carboxamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
ethyl 5-{[benzyl(2-hydroxyethyl)amino]methyl}-1-(4-fluorophenyl)-1H-pyrazole-4-carboxylate
2-(1,3-benzoxazol-2-ylsulfanyl)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}butan-1-one
N-methyl-6-(pyrazin-2-yl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-(3-methoxybenzoyl)-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazine
(1R,6S)-9-methyl-3-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3,9-diazabicyclo[4.2.1]nonane
2-oxo-N-[3-(pyrrolidin-1-yl)propyl]-1,2-dihydroquinoline-4-carboxamide
2-(4,4-difluoropiperidine-1-carbonyl)-1,7-dimethyl-1H-indole
(2R,3R,6R)-5-(3-fluorobenzoyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-[1-(2,2-dimethylpropyl)-4-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N-[3-(5-methyl-4-{[2-(1,3-thiazol-4-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide
4-(1-benzyl-3-methyl-1H-1,2,4-triazol-5-yl)-1-(oxolane-2-carbonyl)piperidine
4-phenyl-N-{1-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
(3S,4S)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(3-methoxyphenyl)piperidin-3-ol
methyl 2-{1-[2-(1H-imidazol-2-yl)benzoyl]-3-oxopiperazin-2-yl}acetate
3-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}pyridin-2-amine
4-(3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-1-phenylpiperazin-2-one
[(6-chloroquinolin-2-yl)methyl](methyl)(oxan-2-ylmethyl)amine
1-{2-[benzyl(methyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}-N,N-dimethylpyrrolidin-3-amine