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N,N-diethyl-3-[({[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}amino)methyl]pyridin-2-amine
N-[(8-methoxyquinolin-2-yl)methyl]-1-(3-phenylpropyl)piperidin-3-amine
(1R,5S,8S)-N-[2-(4-fluorophenoxy)pyridin-3-yl]-8-methoxy-3-azabicyclo[3.2.1]octane-3-carboxamide
2-[1-(2-hydroxybutyl)-5-{4-methyl-3-oxo-1H,2H,3H-pyrazolo[3,4-b]pyridin-6-yl}-1H-1,2,4-triazol-3-yl]acetamide
7-[(2,3-difluorophenyl)methyl]-2-[1-(propan-2-yl)piperidine-4-carbonyl]-2,7-diazaspiro[4.5]decane
1-(1-benzylpiperidin-4-yl)-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
1-(furan-3-carbonyl)-3-(2-phenylethyl)piperidine
N-(3-hydroxypropyl)-3-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-4-carboxamide
N-(3-hydroxyadamantan-1-yl)-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(2,4-difluorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
5-chloro-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
N-tert-butyl-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
1-(4-fluorophenyl)-2-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-3-carboxylic acid
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[(1-phenylcyclohexyl)methyl]acetamide
5-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carbonyl]-3,4-dihydropyrimidin-4-one
1-(cyclohexyloxy)-3-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propan-2-ol
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}cyclopropanamine
4-({[2-(2-fluorophenoxy)pyridin-3-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
[(3-chloro-4,5-dimethoxyphenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-(1,2-oxazol-3-ylmethyl)urea
N-{3-[4-(4-cyclohexylpiperazin-1-yl)piperidin-1-yl]phenyl}-4-phenylbutanamide
N-[(4-chlorophenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-(benzyloxy)-1-(2-methylpropyl)-4-(5-oxopyrrolidine-3-carbonyl)-1,4-diazepan-2-one
2-[4-(2-ethoxyethyl)piperazin-1-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
1-methyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(5-{[4-(5-methylfuran-2-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
N-{[7-fluoro-5-(quinolin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-pyrazole-3-carboxamide
ethyl 1-(3-acetyl-1H-pyrazole-5-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-{[7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-{2-[3-(aminomethyl)pyrrolidin-1-yl]-2-oxoethyl}-1-benzyl-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
N-methyl-4-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzene-1-sulfonamide
[(3R,4R)-1-(3-chloro-2-fluorobenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
5-(azepane-1-carbonyl)-N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(butan-2-yl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-[2-(4-fluorophenoxy)ethyl]-1-[2-(trifluoromethyl)benzoyl]-1,4-diazepan-5-one
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-2-methyl-5-propylpyrimidin-4-amine
N-cyclohexyl-N-methyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
2-[3-(1-benzyl-1H-pyrazol-3-yl)phenyl]pyrazine
4-[2-benzyl-4-(3-methoxyphenyl)-5-oxopiperazin-1-yl]-4-oxobutanamide
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidine
(3S)-3-ethyl-N-(4-phenoxyphenyl)morpholine-4-carboxamide
1-[4-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
N-{1-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N,2-dimethylfuran-3-carboxamide
3-(2-fluorophenyl)-1-methyl-3-(2-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)pyrrolidine-2,5-dione
methyl 4-[(4-carbamoyl-3-chlorophenyl)carbamoyl]piperazine-1-carboxylate
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(1s,4s)-4-aminocyclohexyl]acetamide