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3-chloro-2-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-1H-indole
3-[(3S,4R)-3-(propan-2-yl)-4-[4-(1H-pyrazol-1-yl)butanamido]pyrrolidin-1-yl]propanoic acid
N-(2,2-dimethyloxan-4-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-3-{[(4-fluorophenyl)methyl]sulfanyl}propanamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(oxan-4-yl)piperazin-2-yl}ethan-1-ol
7-methyl-N-(3-methyl-4-pentanamidophenyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-6-methylpyridine-2-carboxamide
1-phenyl-4-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)piperazine
N-[2-(3-fluorophenyl)ethyl]-2-methyl-4-phenylpyrimidine-5-carboxamide
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4-(4-fluorophenyl)oxane-4-carboxamide
1-[(2-{[4-(furan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenyl)methyl]-1H-pyrazole
2-{1-[(4-fluorophenyl)methyl]-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl}ethan-1-ol
N-({5-[(6-methylquinolin-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
3-[(4-methoxyphenyl)methyl]-8-[1-(3-methoxyphenyl)propan-2-yl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3S,4R)-3-cyclopropyl-4-(1-ethyl-1H-pyrazole-3-amido)pyrrolidin-1-yl]propanoic acid
2-[2-(3,4-dimethoxyphenyl)ethyl]-4-[3-(3-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
8-(morpholine-4-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(2-methoxyphenyl)ethyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
N-(2-hydroxyethyl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
2-(ethoxymethyl)-N-[2-(pyridin-3-yloxy)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(2-methylpropanamido)-N-propylbenzamide
5-butyl-4-(2-methyl-1,3-thiazole-4-carbonyl)-1-(3-methylphenyl)piperazin-2-one
N-(4-fluorophenyl)-1-(2-methylbenzoyl)piperidin-3-amine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(methylsulfanyl)ethyl]benzamide
1-(2-methoxyacetyl)-N-[(1R,2R,3R,5S)-2,6,6-trimethylbicyclo[3.1.1]heptan-3-yl]piperidine-4-carboxamide
8-[(2-chlorophenyl)methyl]-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1S)-1-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-3-(methylsulfanyl)propyl]acetamide
4-(2-phenylethyl)-1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-N-[2-(pyridin-4-yl)ethyl]pyrimidin-2-amine
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
3,5,7-trimethyl-N-{3-[(pyridin-3-yl)amino]propyl}-1H-indole-2-carboxamide
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[3-(dimethylsulfamoyl)-5-{[(2-methyl-1H-imidazol-4-yl)methyl]amino}benzoyl]piperidine-3-carboxamide
N-ethyl-2-{4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-1-yl}acetamide
(2S,4R)-1-[4-(benzyloxy)butanoyl]-4-acetamido-N-methylpyrrolidine-2-carboxamide
3-(4-fluorophenyl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-one
2-fluoro-5-{[(2-hydroxyethyl)[(1-methyl-1H-imidazol-2-yl)methyl]carbamoyl]amino}-N-methylbenzamide
2-[5-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
4-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-2-(propan-2-yl)-1,3-oxazole
N-benzyl-N-methyl-1-(oxane-4-carbonyl)piperidin-3-amine
4-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl}-2-(pyridin-4-yl)pyridine
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]pyridine-4-carboxamide
1-(furan-2-carbonyl)-3-(2-methoxybenzoyl)piperidine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-amine
4-[(4-fluorophenyl)methyl]-3-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]piperazin-2-one
{3-[(2,4-difluorophenyl)methyl]-1-(isoquinolin-1-yl)piperidin-3-yl}methanol
2-(5-acetylthiophen-3-yl)-1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-(8-fluoro-4-oxo-1,4-dihydroquinoline-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-(dimethylsulfamoyl)-4-phenoxypiperidine-4-carboxylic acid