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N-[2-(3-fluorophenyl)ethyl]-3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-3-ylmethyl)piperidin-3-yl]propanamide
1-(4-{[(1S)-2-hydroxy-1-phenylethyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(1-benzothiophen-2-ylmethyl)[(4-{2-[4-(furan-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]methylamine
[(3S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(pyridine-2-carbonyl)piperidin-3-yl]methanol
1-(4-fluorophenyl)-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}cyclopropane-1-carboxamide
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-4-(pyrrolidine-1-carbonyl)pyridin-2-amine
N-[3-(1H-imidazol-1-yl)propyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]isoquinoline-1-carboxamide
5-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1H-imidazole-4-carboxylic acid
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-ethyl-N-(2-methylprop-2-en-1-yl)benzamide
4-{4-[(5-hydroxyadamantan-2-yl)amino]piperidin-1-yl}-N-(pyridin-3-ylmethyl)benzamide
N-ethyl-5-(3-fluorophenoxymethyl)-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
1-cyclohexyl-4-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine
1-{[5-(methoxymethyl)furan-2-yl]methyl}-N-methyl-N-(2-phenylethyl)piperidin-3-amine
N-[(2-methylphenyl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
4-[(3,4-dimethoxyphenyl)methyl]-3-{2-oxo-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]ethyl}piperazin-2-one
1-(1-methylazepane-2-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
N,N,5-trimethyl-2-({1-[methyl(pyridin-3-ylmethyl)amino]hex-5-en-2-yl}oxy)pyrimidin-4-amine
2-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}pyrrolidin-3-yl)acetic acid
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-methyl-N-(quinolin-5-ylmethyl)acetamide
methyl 6-(propan-2-yl)-2-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{2-[1-cyclohexyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
N-{[4-methoxy-3-(thiophen-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-(4-chloro-2-fluorobenzoyl)-N-(4-methoxyphenyl)piperidin-3-amine
1-{4-[2-(furan-3-yl)-1H-imidazol-1-yl]phenyl}-5-methylpyrrolidin-2-one
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[(2-phenoxypyridin-3-yl)methyl]pyrazine-2-carboxamide
1-ethyl-4-{[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-1H-pyrrole-2-carbonitrile
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(3-fluoropyridin-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(2-methoxyethyl)-2-[(5-methylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decane
N-tert-butyl-3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
7-methyl-2-(3-methylphenyl)-3-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}quinoline
methyl(3-methylbutyl){[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
(4aS,8aR)-2-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}-decahydroisoquinoline
1-(cyclopropylmethyl)-4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-pyrazole
9-[2-(3-fluorophenyl)acetyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(4-{[2-(2-aminoethyl)morpholin-4-yl]methyl}phenyl)-6-butyl-3,4-dihydropyrimidin-4-one
(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]{[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
1-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-4-methoxybenzamide
1-methyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]azepane-2-carboxamide
5-methyl-N-(oxolan-2-ylmethyl)-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)thiophene-2-carboxamide
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
N-ethyl-6-({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-N-methylpyridine-3-carboxamide
N-[5-(2-methylphenyl)-1,3,4-thiadiazol-2-yl]-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
5-acetamido-1-(2-methoxyethyl)-N-[(1S)-1-phenylethyl]-2-(pyridin-2-yl)-1H-1,3-benzodiazole-7-carboxamide
3-methyl-1-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}piperazine
N-[(3S,5S)-1-(cyclopentylmethyl)-5-(diethylcarbamoyl)pyrrolidin-3-yl]pyridine-3-carboxamide