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1-[(diethylcarbamoyl)methyl]-N-methyl-N-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]benzonitrile
(1R,5R)-6-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
6-(azepan-1-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-(morpholin-4-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
methyl 4-[4-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperazin-1-yl]benzoate
N-[(2R,3R)-1'-[(2-hydroxy-4-methoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
ethyl 2-[2-({1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazol-4-yl}formamido)ethyl]-1,3-thiazole-4-carboxylate
(3S)-3-{[5-(4-chlorophenyl)-1,2,4-triazin-3-yl]amino}azepan-2-one
3-(3-methylphenyl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidine
4-(4-{[(3-chlorophenyl)methyl]amino}piperidin-1-yl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
3-(1-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
(4aS,7aR)-1-[2-(3-chlorophenyl)acetyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,4-dimethylbenzamide
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-propyl-1,3-thiazole-4-carboxamide
4-[(2R)-2-hydroxy-2-phenylacetyl]-1-(2-methoxyphenyl)piperazin-2-one
1-cyclopropyl-3-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-methylbutanamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2-methoxyphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
1-[(2-fluorophenyl)methyl]-N-[1-(3-methoxyphenyl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-(2-methoxyethyl)-3-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]propanamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(pyridin-3-ylmethyl)piperidin-4-yl]oxy}benzamide
methyl 1-[9-methoxy-7-oxo-3-(3-phenylpropyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]piperidine-2-carboxylate
N-(4-fluoro-2-methylphenyl)-3-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-yl]propanamide
(3R,5S)-N-butyl-5-(morpholin-4-ylmethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
2,3-dimethyl-N-[1-(thian-4-yl)piperidin-4-yl]-1H-indole-5-carboxamide
5-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
N-cyclopropyl-2-(dimethylamino)-2-(3-methylphenyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-N,5-dimethyl-N-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluorobenzamide
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(pyridin-3-yl)ethan-1-one
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
(5S,9aS,9bS)-2-methyl-5-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-7,8-dimethyl-3,4-dihydroquinazolin-4-one
5-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
N-[3-(1,3-oxazol-5-yl)phenyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
1-methyl-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)azepane-2-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-methoxy-5-oxo-6-pentyl-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
6-(1-methyl-1H-imidazol-2-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyridazin-3-amine
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
{2-oxo-2-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]ethyl}urea
4-{[1-(2H-1,3-benzodioxol-5-yl)-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
1-ethyl-5-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrrolidine-3-carboxamide
1-{2-[1-(2-methoxyphenyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidine