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N-cycloheptyl-3-[4-(prop-2-en-1-yl)piperazin-1-yl]propanamide
2-{1-[(2-butyl-1H-imidazol-4-yl)methyl]pyrrolidin-2-yl}-1,3-benzothiazole
(1S,6R)-3-[(2-fluoro-4-methoxyphenyl)methyl]-3,9-diazabicyclo[4.2.1]nonane
1-{2-[5-(1H-indol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
3-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-ol
2-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(4-methylphenoxy)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]piperidine-4-carboxamide
1-methyl-3-(propan-2-yl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1H-pyrazole-5-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(3-hydroxy-3-methylbutyl)benzamide
4-[3-(3-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}phenoxy)propyl]morpholine
N-(1-{7-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)pyridine-3-carboxamide
methyl 4-[({[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}amino)methyl]benzoate
3-(oxolan-3-yl)-2,4,5-triazatetracyclo[11.4.0.02,6.07,12]heptadeca-1(17),3,5,7,9,11,13,15-octaene
12-(4-hydroxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
3-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
N-{[4-(2H-1,3-benzodioxol-5-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl}-N-methylmethanesulfonamide
1-[2-(4-fluorophenyl)ethyl]-4-[(1-propylpiperidin-4-yl)amino]pyrrolidin-2-one
5-(1-benzofuran-2-yl)-3-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-1,2,4-triazine
N1-[4-(pyridin-2-ylmethoxy)phenyl]piperidine-1,4-dicarboxamide
1-(3-phenylpropyl)-4-(pyrazin-2-yl)-1,4-diazepane
N-{3-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-3-oxopropyl}-N-methylmethanesulfonamide
N-(1-benzothiophen-5-ylmethyl)-2-(4-oxo-1,4-dihydropyridin-1-yl)acetamide
1-(6-ethylpyrimidin-4-yl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
1-[(3-chlorophenyl)methyl]-4-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperazine
4-{2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]acetyl}-1-cyclopentylpiperazin-2-one
5-ethyl-N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-[(3R,4S)-1-(morpholine-4-sulfonyl)-4-propylpyrrolidin-3-yl]pyrimidin-2-amine
2-methyl-5-[(3-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}-1,2-oxazol-5-yl)methoxy]pyridine
N-cyclopropyl-3-{[(2-methanesulfonamidoethyl)carbamoyl]amino}-4-methoxybenzamide
6-methoxy-1-[(4-methoxyphenyl)methyl]-4-[5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carbonyl]-1,4-diazepan-2-one
2-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
1-{3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanoyl}-1,4-diazepan-5-one
1-cyclopentyl-4-[5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carbonyl]piperazin-2-one
5-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}-2-(3-methylphenyl)pyrimidine
{2-[4-(2-chlorophenoxy)piperidin-1-yl]quinolin-3-yl}methanol
2-{[(2-methoxy-6-methylphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-{3-[3-(benzyloxy)azetidine-1-carbonyl]piperidin-1-yl}acetamide
3-amino-1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]propan-1-one
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(5-methyl-2-phenylfuran-3-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
2-(2,6-dichloropyridin-4-yl)-6-(1-methylpiperidin-3-yl)-3,4-dihydropyrimidin-4-one
4,4,4-trifluoro-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}butanamide
10-methoxy-5-[2-(2-methoxyphenoxy)ethyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
3,4,4-trimethyl-1-(3-phenyl-1,2-oxazole-5-carbonyl)pyrrolidin-3-ol
2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N,N-bis(prop-2-en-1-yl)acetamide
3-{[(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)amino]methyl}pyrrolidin-3-ol
5-[3-(1,3,4-oxadiazol-2-yl)phenoxy]-1-azabicyclo[3.2.1]octane
N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-2-methyl-1H-1,3-benzodiazole-5-carboxamide
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-2-ylsulfanyl)acetamide
2,7-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-5-carboxamide