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1-{4-[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(2-methoxyphenyl)ethan-1-one
2-[3-(4-methoxyphenyl)-1-(3-methylbutyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
(2R,6R)-4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-{[3-(4-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}-4-(methylsulfanyl)butanoic acid
N-(furan-2-ylmethyl)-4-{[4-(2-hydroxypropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
2-(1,2-benzoxazol-3-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
methyl 3-{methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]carbamoyl}propanoate
9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-4-(2-methoxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl (2S)-3-(1H-imidazol-4-yl)-2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propanoate
butyl 9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxylate
3-({1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
N-({3-methyl-7-[2-(thiophen-2-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
5-{1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1H-1,2,3-triazol-4-yl}pyrimidine
1-ethyl-N-[(2S)-1-hydroxybutan-2-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-1,2-oxazole-3-carboxamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-(cycloheptylamino)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxylic acid
1-[(2-chlorophenyl)methyl]-N-(1-methoxypropan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-ethyl-2-(morpholin-2-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
2-methoxy-2-phenyl-N-(1-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
3-{2-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-(2-methoxyethyl)-5-{4-phenyl-1-[3-(pyridin-4-yl)propyl]-1H-imidazol-5-yl}pyrimidine
N-[(2S,4R,6S)-2-(2-butoxy-3-methoxyphenyl)-6-ethyloxan-4-yl]acetamide
ethyl 2-{N-methyl-1-[6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridin-3-yl]formamido}acetate
N-[2-(3-methoxyphenyl)-1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
3-(2-chloro-4-fluorobenzenesulfonyl)-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
(4aS,8aR)-6-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
(1S,2S)-2-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}cyclohexan-1-ol
6-[(3,3-dimethylcyclohexyl)amino]-2-methylheptan-2-ol
N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-4H-chromene-2-carboxamide
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
N-({3-methyl-7-[4-(thiophen-2-yl)butanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)pyrazine-2-carboxamide
(2S,4S)-4-amino-N-{[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methylpyrrolidine-2-carboxamide
2-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
N-ethyl-2-(2-methylphenyl)-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}acetamide
2-(2-methoxyethyl)-6-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1,3-benzoxazole
(1R,3s,6r,8S)-4-{5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carbonyl}-4-azatricyclo[4.3.1.13,8]undecane
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]butanamide
2-(dimethylamino)-N-(2-acetamidoethyl)-2-(2-methylphenyl)acetamide
methyl[1-(3-methylpyridin-2-yl)propan-2-yl]{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyrimidin-4-amine
(1S,4S)-2-(2-fluorophenyl)-5-(quinoxalin-5-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-[(4-fluorophenyl)methyl]-5-methyl-5-{1-[1-(piperidin-1-yl)cyclohexanecarbonyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[(5-methylpyrazin-2-yl)methyl]-4-(piperidin-3-yl)benzamide
3-{1-[4-(piperidin-1-yl)benzoyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-[(4-fluorophenyl)methyl]-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
6-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
3-(1-methyl-1H-imidazol-2-yl)-6-[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyridazine
(1S,5R)-N-(2,4-dimethoxyphenyl)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide