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3-[3-(4-ethylpiperazin-1-yl)propyl]-8-[(2R)-2-hydroxypropanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-(4-ethylpiperazin-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-[(1S)-2,3-dihydro-1H-inden-1-yl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
7-fluoro-2-methyl-4-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinoline
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
(5-{1-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
2-chloro-4-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}phenol
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
1-[2-(1H-imidazol-1-yl)ethyl]-4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazine
2-(ethylamino)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)pyrimidine-5-carboxamide
N-ethyl-N-[(5-methylfuran-2-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-[3-(5-methylfuran-2-yl)-5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-1H-1,2,4-triazol-1-yl]butan-2-ol
2-(1-{3-[(5-methylpyridin-2-yl)amino]propyl}-1H-imidazol-2-yl)benzoic acid
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-methyl-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(pyrimidin-4-ylmethyl)-1,2-oxazole-3-carboxamide
5-methyl-4-{methyl[2-(4-methylphenoxy)ethyl]amino}-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
3-[5-(1-benzothiophen-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
2-methyl-4-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
4-ethyl-1-methyl-3-[1-(3-methyl-1H-indole-2-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-ethyl-1H-pyrazol-5-yl)-1-(2-phenylpropyl)piperidine
5-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-(4-acetylphenoxymethyl)-N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-1,2-oxazole-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(phenylamino)pyrimidine-5-carboxamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)acetamide
5-(2-{2-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
1-[(3S,4R)-1-[2-(2-chloro-4-fluorophenyl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
2-amino-6-(4-chlorophenyl)-4-(furan-3-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-4-(pyrrolidin-1-ylmethyl)benzamide
N-[4-(1H-indol-2-yl)phenyl]-1-(pyridine-4-carbonyl)piperidine-4-carboxamide
2-{[(4aS,7aR)-4-(2-hydroxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
5-(2H-1,3-benzodioxol-5-yl)-3-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-1,2,4-triazine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propanamide
N-butyl-2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-methylacetamide
2-{4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl}acetic acid
5-(1H-imidazol-1-ylmethyl)-2-[4-(3-methylphenoxy)piperidin-1-yl]pyridine
N-benzyl-5-[(3,4-difluorophenyl)methyl]-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(5-{[(3S)-3-(dimethylamino)azepan-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
methyl 1-[(3S,5S)-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
8-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}quinoline
N-(3-ethoxy-2-hydroxypropyl)-N'-(4-methylphenyl)propanediamide
1-benzyl-5-methanesulfonamido-2-methyl-N-[(2-methylphenyl)methyl]-1H-1,3-benzodiazole-7-carboxamide
3-(2-chlorophenyl)-N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-3-phenylpropanamide
ethyl 4-(3-phenylpropyl)-1-(prop-2-ene-1-sulfonyl)piperidine-4-carboxylate
1-[(3,4-dimethoxyphenyl)methyl]-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
N-cyclopropyl-3-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)propanamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-(pyrazin-2-ylmethyl)acetamide