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1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4-(1H-pyrazol-1-yl)butan-1-one
7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-4-(1-propylpiperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,3S)-3-methoxy-7-[4-methoxy-3-(prop-2-en-1-yl)benzoyl]-3-methyl-7-azaspiro[3.5]nonan-1-ol
1-methyl-5-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-imidazole
2-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)-1H-1,3-benzodiazole
(1R,5R)-6-benzyl-3-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
9-methoxy-7-(4-methoxyphenyl)-4-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{2-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-(methanesulfonylmethyl)-1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidine
4-chloro-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(furan-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3,5-difluorophenyl)-4-[(2-ethyl-1H-imidazol-1-yl)methyl]-5-methyl-1,3-oxazole
N-butyl-2-[(dimethylcarbamoyl)amino]-N-[(4-fluorophenyl)methyl]acetamide
8-(1-benzofuran-5-ylmethyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[benzyl({[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl})amino]ethan-1-ol
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
N-[(5-methylfuran-2-yl)methyl]-3-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-yl]propanamide
1-cyclopentanecarbonyl-4-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]piperidine
2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-8-methoxyquinoline
14-[2-(1H-pyrazol-1-ylmethyl)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[(2-methoxyphenyl)methyl]-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
6-{[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]methyl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-cyclopentyl-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
5-(methoxymethyl)-N-(3-methyl-1-{7-[(2E)-4-methylpent-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
(5S,9aS,9bS)-5-(4-methoxynaphthalen-1-yl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(2R,3R)-1'-(2-oxo-2-phenylacetyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
methyl[3-(oxolan-2-yl)propyl]{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
2-(2-phenylethyl)-5-(thiomorpholine-4-carbonyl)-1,3-benzoxazole
5-cyclopropyl-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,3,4-oxadiazol-2-amine
9-[2-(ethylsulfanyl)propanoyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(4-methylphenyl)acetamide
7-[(3,4-difluorophenyl)methyl]-2-(5-methyl-1,2-oxazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methyl-1-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]urea
2-[(2-chlorophenyl)methyl]-4-[3-(2-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(pyrrolidine-1-sulfonyl)thiophene-2-carboxamide
1,1,1-trifluoro-3-{2-[4-methoxy-3-(methoxymethyl)phenyl]-1H-imidazol-1-yl}propan-2-ol
2-(4-fluorophenyl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}acetamide
N-cyclopropyl-4-methoxy-3-({1-[1-(3-methylpyridin-2-yl)propan-2-yl]piperidin-4-yl}oxy)benzamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-(morpholin-4-yl)benzamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[2-(phenylsulfanyl)ethyl]acetamide
3-{[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](methyl)amino}propane-1,2-diol
methyl 5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(oxane-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-(1H-1,3-benzodiazol-1-yl)-1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(pyridine-4-carbonyl)-1,4-diazepan-2-one