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1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(piperidin-1-yl)piperidine-4-carboxamide
2-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
(1S,5R)-3-[1-(3-chlorophenyl)piperidin-4-yl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
3-{1-[6-(dimethylamino)pyrimidin-4-yl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-phenylcyclopropane-1-carboxamide
(4aS,7aR)-1-pentanoyl-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(2-methoxyphenyl)ethyl]-6-(quinoxalin-5-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridine
N-(pyridin-2-ylmethyl)-5-{spiro[2.3]hexane-1-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
3-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1-[3,5-difluoro-4-(trifluoromethyl)phenyl]-3-methylurea
N-(2-methoxyethyl)-2-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinoline-8-sulfonamide
4-[1-ethyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]butanoic acid
2-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(pyrrolidin-1-yl)pyrazine
1-[1-(furan-2-yl)ethyl]-2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazole
2-{3-cyclopropyl-5-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]-1H-1,2,4-triazol-1-yl}pyridine
4-{5-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
3-cyclopropyl-5-(2-methoxyphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
2-{1-[2-(dimethylamino)ethyl]-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl}-N-methyl-N-[3-(piperidin-1-yl)propyl]acetamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-4-phenylbenzamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-amino-6-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]pyrimidin-4-ol
(4R)-N,3-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,3-thiazolidine-4-carboxamide
7-[4-(3-hydroxypiperidin-1-yl)piperidine-1-carbonyl]quinolin-8-ol
3-(2,4-dimethoxybenzoyl)-1-[(2,3,6-trifluorophenyl)methyl]piperidine
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)methanesulfonamide
3-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]urea
methyl 2-{[7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]sulfonyl}benzoate
(1R,2R)-N-methyl-2-phenyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]cyclopropane-1-carboxamide
N-(4-methoxy-2-methylphenyl)-3-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-3-yl}propanamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
2-ethyl-7-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
6-(benzyloxy)-1-(2-methylpropyl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-2-one
9-(6-methylpyrimidin-4-yl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[7-(4-ethenylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}propane-1-sulfonamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-fluoroethyl)-5-methoxybenzamide
2-(4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
4-(7-chloro-1-methyl-1H-indole-2-carbonyl)-1,4-oxazepan-6-ol
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}furan-3-carboxamide
1-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]pyrrolidin-2-one
N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-2-(trifluoromethyl)benzene-1-sulfonamide
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
1-ethyl-5-({[(2-fluoro-4-methylphenyl)carbamoyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(quinolin-6-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-chloro-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole
N-[(1-benzylpyrrolidin-3-yl)methyl]-3-methylpyrazin-2-amine
4-({5-[2-(thiophen-2-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)piperazin-2-one
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]propanamide