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N-[2-(2-chloro-6-fluorophenyl)ethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]-3-methylbut-2-en-1-one
1-[1'-(1-benzothiophen-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-{4-[4-(4-methoxyphenoxy)piperidin-1-yl]-4-oxobutyl}piperidin-2-one
(4aS,7aR)-1-(pyridine-4-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(diethylamino)ethyl]-N-ethyl-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
2-(4-methoxyphenyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)acetamide
1-[4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-4-(2-methylpropyl)-1,4-diazepane
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(2-methoxyethyl)methylamine
N-({5,7-dimethylimidazo[1,2-a]pyridin-2-yl}methyl)-5-methoxy-1-methyl-1H-indole-2-carboxamide
N-[1-(4-fluorophenyl)ethyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-[(3S,4R)-1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
(2S,4S)-N-ethyl-1-(propan-2-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-methyl-4-(4-{[4-(piperazin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyrimidine
3-(4-chlorophenyl)-N-methyl-3-phenyl-N-(pyridin-3-ylmethyl)propanamide
N-[(4-chlorophenyl)(phenyl)methyl]-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
8-chloro-2-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]quinoline-4-carboxamide
1-[1-ethyl-5-(5-ethyl-1,2-oxazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1,1-dioxo-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
3-cyclopropyl-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1H-pyrazole-5-carboxamide
methyl 1-benzyl-3-cyclopropaneamido-5-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(5-ethylpyridin-2-yl)methyl]-3-(2-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
(1R,9aR)-1-{[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}-octahydro-1H-quinolizin-1-ol
1-(2-ethoxyethyl)-4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperazine
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-2-yl)piperazine
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-{[(4-fluorophenyl)methyl](methyl)amino}ethan-1-one
1-[4-(3-methyl-3-phenylpiperidine-1-carbonyl)phenyl]imidazolidine-2,4-dione
3-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2-oxazole-5-carboxamide
3-({[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
ethyl 1-[(4-hydroxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
3-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N,N-dimethylpyrazin-2-amine
1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-4-(1H-imidazol-2-ylmethyl)-1,4-diazepan-6-ol
9-(4-chloro-1H-pyrazole-3-carbonyl)-3-methyl-3,9-diazaspiro[5.6]dodecane
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
4-[2-(propan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine
3-methoxy-N-[1-(7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]propanamide
3-oxo-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-3,4-dihydroquinoxaline-2-carboxamide
2-[3-(5-methylfuran-2-yl)-5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
N-(1,2-oxazol-3-ylmethyl)-2-(phenylamino)pyrimidine-5-carboxamide
6-methoxy-3-methyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1-benzofuran-2-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-(5-propylpyrimidin-4-yl)pyrrolidine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2,4-dioxoimidazolidin-1-yl)-N-[(4-methylphenyl)methyl]acetamide
2-{4-[1-(2,3-dimethylphenyl)piperidin-4-yl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(2,2,6-trimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)acetamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
ethyl 2-{1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]piperidin-2-yl}acetate
1-(2-methylpropyl)-4-(1-phenylmethanesulfonylpyrrolidin-3-yl)piperidine
6-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-N,N-dimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-2-(propan-2-yl)oxane-4-carboxamide