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N-{4-[4-({[3-(dimethylamino)phenyl]formamido}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}-5-(methoxymethyl)furan-2-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-5-[(methylsulfanyl)methyl]furan-2-carboxamide
(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(3S,5R)-1-[(2-methylphenyl)methyl]-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-(2,1,3-benzothiadiazol-4-ylmethyl)-1-(carbamoylmethyl)piperidine-3-carboxamide
N-[(2R,3R)-1'-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-(3-{[4-(3-fluorophenoxy)piperidin-1-yl]methyl}phenyl)ethan-1-amine
2-{[1-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,2-dihydrophthalazin-1-one
(4aS,7aR)-1-[(4-acetylphenyl)methyl]-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)methanesulfonamide
5-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-butyl-5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-1H-1,2,4-triazole
methyl 3-(2-methoxyacetamido)-1-(3-methylbutyl)-5-[(2-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,2-dimethyl-6-(piperidin-4-yl)pyrimidin-4-amine
4-(1,3-benzothiazol-2-yl)-2-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenol
5-(4-chloro-2-methoxyphenoxymethyl)-3-(pyrrolidine-1-carbonyl)-1,2-oxazole
7-(2,2-dimethylpropyl)-2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
8-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(1-benzothiophen-5-ylmethyl)-4-ethyl-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
N-(2-hydroxyethyl)-8-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
(2S,4R)-N-(2-methoxyethyl)-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
3,5-dimethyl-1-(1-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}pyrrolidin-3-yl)-1H-pyrazole
3-ethoxy-1-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
3-methoxy-N-[1-(7-{[4-(methylsulfanyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]propanamide
3,4,7-trimethyl-2-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-1H-indole
(5S,9aS,9bS)-5-[4-(dimethylamino)phenyl]-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-2-(2-ethoxyphenyl)ethan-1-one
N-[2-(4-fluorophenoxy)ethyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-(2-methoxy-5-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-{1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-phenyl-1,3-thiazole-2-carboxamide
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N-[2-(3,4-dimethoxyphenyl)ethyl]-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}acetamide
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)pent-4-enamide
{[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
5-(2-methoxyacetamido)-1-methyl-N-(oxolan-2-ylmethyl)-N-propyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
3-{2-[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-(4-fluorophenyl)-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-amine
1-[3-(3,4-dimethoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4-(piperidin-1-yl)piperidine
(1R,2R,4R)-N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(pyridin-3-ylmethyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-7,8-dimethyl-2-(pyrimidin-5-yl)quinoline
5-(5-methylfuran-2-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1,2,4-triazin-3-amine
4-(3,5-dimethyl-1H-indole-2-carbonyl)-1λ6-thiomorpholine-1,1-dione
1-[1'-(3-propyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-(pyrrolidin-3-yl)ethan-1-one
1-(1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
2-{2-[4-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)piperazin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
4-(1-butyl-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine