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methyl 6-[(3-hydroxyphenyl)methyl]-2-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[(4aS,7aR)-4-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzene-1-sulfonamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperazine
1-phenyl-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
ethyl 4-(1-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperidin-3-yl)piperazine-1-carboxylate
N-(5-chloro-2-methoxyphenyl)-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)propanamide
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-4-oxo-3,4-dihydrophthalazine-1-carboxamide
[(4-fluoro-2-methoxyphenyl)methyl]({[2-(morpholin-4-yl)pyridin-3-yl]methyl})amine
1-cyclohexyl-4-oxo-N-[phenyl(pyridin-4-yl)methyl]-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-(1H-imidazol-2-yl)-N-(2-methylquinolin-4-yl)benzamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-({7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-fluorobenzamide
2-benzoyl-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-tert-butyl-4-[4-hydroxy-4-(pyridin-3-yl)piperidine-1-carbonyl]pyrrolidin-2-one
({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)(methyl)[(5-methylfuran-2-yl)methyl]amine
2-(4-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}phenyl)ethan-1-amine
methyl 3-(2-chloro-6-fluorobenzamido)-6-{[(2-methoxyethyl)(methyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
3-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-(1,3-thiazol-4-ylmethyl)piperidine
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(5-methyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methanol
N-({7-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-methoxy-2-phenylacetamide
{1-[1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanamine
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(quinoxalin-2-ylmethyl)benzamide
(3R,4R)-1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
5-ethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-(3-methoxypropanoyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl]({[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})(pyridin-3-ylmethyl)amine
3-(pyridin-3-yl)-N-({7-[(2,3,4-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)propanamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)pyridine-4-carboxamide
N-{2-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-methoxybenzamide
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2,4-dimethyl-N-(4-{4-[(pyridin-3-ylmethyl)amino]piperidin-1-yl}phenyl)benzamide
2-[5-(1-ethyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-phenylethan-1-ol
5-(2-methoxyethyl)-3-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
N-cyclopropyl-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}-3-(hydroxymethyl)pyrrolidin-3-ol
1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1-(pyridin-4-ylmethyl)urea
N-[3-(4-fluorophenyl)phenyl]-1-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
4-({4-methyl-5-[1-(pyrimidin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
8-(1-methyl-1H-pyrrole-2-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
1-(7-methoxy-4-methylquinazolin-2-yl)-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]oxy}benzamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(2-oxoazepan-1-yl)acetamide
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-(1H-indol-6-ylmethyl)piperidin-4-amine
2-{[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzoic acid
3-[(4-cyclohexylpiperazin-1-yl)methyl]-1-[2-(dimethylamino)ethyl]-7-methyl-1,2-dihydroquinolin-2-one
3-{1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
8-(2,2-dimethylpropyl)-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[4-(pyridin-4-yl)piperidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine