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2-[1-cyclopropyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-5-(3-fluorophenoxymethyl)-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-3-carboxamide
6-fluoro-4-[2-(4-methylpentyl)morpholine-4-carbonyl]-1,2-dihydroquinolin-2-one
3-(dimethoxy-1,3,5-triazin-2-yl)-4H-chromen-4-one
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-methyl-N-(2-{2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)methanesulfonamide
4-[2-(dimethylamino)benzoyl]-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
5-(dimethylamino)-2-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-2,3-dihydropyridazin-3-one
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-N-(4-methoxy-2-methylphenyl)piperidine-1-carboxamide
5-benzyl-5-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
5-{2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-fluoro-3-[2-(3-methoxyphenyl)azetidine-1-carbonyl]benzene-1-sulfonamide
1-(azocan-1-yl)-3-[2-methoxy-4-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N4-cyclopropylpyrimidine-2,4-diamine
2-methyl-1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-(4-methylphenyl)piperazine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)[3-(5-methylfuran-2-yl)butyl]amine
1-(2,3-dihydro-1-benzofuran-2-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
4-(2-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-2-yl}ethyl)morpholine
N-(3-chlorophenyl)-2-[2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]acetamide
4-{5-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperazin-2-one
2-(3-fluoro-4-hydroxyphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]acetamide
(5-{[ethyl(oxan-4-ylmethyl)amino]methyl}furan-2-yl)methanol
N-(3-ethoxy-2-hydroxypropyl)-1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
8-(2-ethoxybenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
4-[(4-methoxy-3-methylphenyl)methyl]-3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
5-[(5-chloro-2,3-dimethoxyphenyl)methyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]amino}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(furan-2-ylmethyl)-9-methoxy-3-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
methyl 4-{[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]methyl}benzoate
4-[2-(4-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethyl]morpholine
ethyl 4-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]piperazine-1-carboxylate
N-(1-{7-[(9-ethyl-9H-carbazol-3-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
6-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
4-phenyl-3-{1-[2-(1,2,3,6-tetrahydropyridin-4-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(furan-3-ylmethyl)(methyl)[4-(morpholin-4-yl)butyl]amine
2-(1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
9-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1'-(3,4-difluorobenzoyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-(4-cyclohexylpiperazine-1-carbonyl)-2-(propan-2-yl)-1,3-benzoxazole
methyl 7-oxo-9-[3-(pyridin-4-yl)propoxy]-3-(thiophene-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
4-{4-[2-(2-chlorophenyl)-2-hydroxyacetyl]piperazin-1-yl}-2-(naphthalen-1-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(pyrazine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-chloro-3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinolin-4-ol
2-(5-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl)pyridine