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(1R)-2-{3-[3-(6-methoxypyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}-1-phenylethan-1-ol
ethyl 4-(2-methoxyethyl)-1-[2-(3-methylphenyl)benzoyl]piperidine-4-carboxylate
1-[2-oxo-2-(3-propoxypiperidin-1-yl)ethyl]-1,2,3,4,5,6,7,8-octahydroquinolin-2-one
N,N-diethyl-1-{[2-hydroxy-5-(6-methoxypyridin-2-yl)phenyl]methyl}piperidine-3-carboxamide
2-{1-[(2-fluorophenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
(2E)-3-(3-fluorophenyl)-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)prop-2-enamide
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-3-(2-oxopyrrolidin-1-yl)benzamide
3-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]benzonitrile
ethyl 4-[4-(4-{[(3-chlorophenyl)methyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
(3R)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-N-{[3-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
1-cyclohexyl-N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(4aS,8aR)-6-(2-hydroxy-3-methylbenzoyl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-1-methylpyrrolidine-3-carboxamide
2-(methoxymethyl)-5-{[4-(4-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine
1-cycloheptyl-N-[(2-methylpyridin-4-yl)methyl]-6-oxopiperidine-3-carboxamide
2,2-dimethyl-3-{[1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propan-1-ol
methyl 3-(2-methyl-1H-imidazol-4-yl)benzoate
1-(furan-2-ylmethyl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
N-[(3-fluorophenyl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-methyl-5-[methyl(naphthalen-1-ylmethyl)amino]-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(furan-2-ylmethyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N,3-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-oxo-3,4-dihydrophthalazine-1-carboxamide
5-ethyl-5-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
3-(1H-1,2,3-benzotriazol-1-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one
8-(5-chloro-2-fluorobenzoyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-(3-chlorophenyl)-N-[1-(pyridin-4-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N-[2-(cyclohexylsulfanyl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
3-(2-{3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
N-(3-chloro-4-fluorophenyl)-3-[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-4-yl]propanamide
N-(3,4-dimethoxyphenyl)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-3-amine
7-[(3,5-dimethylphenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N,8-dimethyl-N-(1-methylpiperidin-4-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
(4aS,7aR)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-3-(pyridin-3-yl)propan-1-one
2-methoxy-N-{[3-(methylsulfanyl)phenyl]methyl}-N-(propan-2-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
2-(1-{[1-(thiophene-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[(2-methyl-1H-indol-5-yl)methyl]amine
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-(propan-2-yl)pyrimidin-4-amine
3-ethyl-1-methyl-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-1H-pyrazole-5-carboxamide
5-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-4-methylpyrimidin-2-amine
1-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-ethylurea
1-(2-chloropyridin-3-yl)-3-[2-(dimethylamino)ethyl]-3-[(3-methylthiophen-2-yl)methyl]urea
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-{3-[benzyl(methyl)amino]piperidin-1-yl}ethan-1-one
N-cyclopentyl-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(prop-2-en-1-yl)acetamide
4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N-methyl-1,3-thiazol-2-amine