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6-methoxy-3-methyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-1-benzofuran-2-carboxamide
4-[5-methyl-4-(thiophen-2-yl)-1H-imidazol-2-yl]-1-[(4-methylphenyl)methyl]pyrrolidin-2-one
1-cyclohexyl-4-oxo-N-[(4-phenyloxan-4-yl)methyl]-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-methoxy-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)benzamide
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-2-oxo-1,4-diazepan-6-yl}oxy)acetamide
5-[2-(phenylamino)pyrimidine-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
6-ethyl-4-[2-(4-fluorophenyl)morpholine-4-carbonyl]-1,2-dihydropyridin-2-one
1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3-cyclopentylpropyl)-N-methyl-1,2,5-oxadiazole-3-carboxamide
N-[2-(dimethylamino)ethyl]-3-(1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)propanamide
2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-3-(4-propylpiperazine-1-carbonyl)-1,4-dihydropyridin-4-one
2-[4-(1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)morpholin-3-yl]acetamide
2-(dimethylamino)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-2-(4-methylphenyl)acetamide
4-cyclopentyl-3-(3-hydroxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[1-(2-methoxyethyl)piperidin-3-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
1-[(1-hydroxycyclohexyl)methyl]-3-(6-phenoxypyridin-3-yl)urea
1-{3-[(E)-2-phenylethenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-(thiophen-2-yl)propan-1-one
5-(2-methyl-1,3-thiazole-4-carbonyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[(1-ethyl-1H-indol-4-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
{1-[(2-chloro-4-fluorophenyl)methyl]-3-[(4-fluorophenyl)methyl]piperidin-3-yl}methanol
4-{4-[4-(cyclopropylmethyl)piperazine-1-carbonyl]phenoxy}-N,N-dimethylpiperidine-1-sulfonamide
4-(1-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}piperidine-4-carbonyl)morpholine
1-(2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-1H-pyrazole
3-(2-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
methyl 3-[(2-fluoro-5-methoxyphenyl)methyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
N,N-bis(2-hydroxyethyl)-2-methyl-4-oxo-1,4-dihydroquinoline-8-carboxamide
(5S,9aS,9bS)-2-methyl-5-(2,4,6-trimethoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
9-{[3-(butan-2-yloxy)phenyl]methyl}-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
2-[(oxolan-3-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
6-methyl-2-oxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2-dihydropyridine-4-carboxamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-2-[4-(3-methylphenyl)piperazin-1-yl]acetamide
4-[2-(dimethylamino)-2-(4-methylphenyl)acetamido]-N,N-dimethylbutanamide
N-[(4-methoxyphenyl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
(2S,4S)-4-{[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]amino}-N-ethyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methylacetamide
6,8-dimethyl-2-({[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]amino}methyl)quinolin-4-ol
2-(methoxymethyl)-N,1-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-(2-phenylacetamido)-1H-1,3-benzodiazole-7-carboxamide
1-(2-methoxyethyl)-3-methyl-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3,4-dimethylphenyl)-1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}propan-1-one
methyl 4-{4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperazin-1-yl}benzoate
2-[3-(2-aminoethyl)piperidine-1-carbonyl]-N-[(3-methylthiophen-2-yl)methyl]aniline
2,2-dimethyl-1-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-4-yl]-5-ethylimidazolidine-2,4-dione
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(methylsulfanyl)pyrimidin-4-amine
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-yl)acetamide
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol