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5-(dimethylamino)-2-{2-[4-(morpholine-4-carbonyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
3-({1-[3-(2,3-dihydro-1H-indol-1-yl)propanoyl]pyrrolidin-3-yl}methyl)benzamide
1-(2-methylbenzoyl)-4-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]piperidine
3-{benzyl[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}-2-methylpropan-1-ol
4-[(4-fluorophenyl)methyl]-1-(1,3-thiazol-4-ylmethyl)piperidine
1-tert-butyl-4-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}pyrrolidin-2-one
3-(4-methoxyphenyl)-1-methyl-3-[2-oxo-2-(3-propanoylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione
(3R,4R)-3-cyclobutyl-4-methyl-1-(1-phenylcyclopropanecarbonyl)pyrrolidin-3-ol
N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-[(propan-2-yl)amino]benzamide
(2R)-1-({2-[butyl(methyl)carbamoyl]imidazo[1,2-a]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
2-[3,5-dimethyl-4-(pyridin-4-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
5-{1-[(1S)-1-(3-methoxyphenyl)ethyl]-1H-imidazol-2-yl}-4-methyl-1H-imidazole
methyl (2S)-1-({4-[(2-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)pyrrolidine-2-carboxylate
(2E)-3-(2-chlorophenyl)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)prop-2-enamide
2-[(3-chlorophenyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(2-{[(3-methoxyphenyl)methyl]carbamoyl}ethyl)-N-(2-phenylethyl)piperidine-1-carboxamide
(3R,4S)-4-cyclopropyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidin-3-amine
1-(2-chloro-3,5-difluorophenyl)-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
7-({[(2-fluorophenyl)methyl](2-methoxyethyl)amino}methyl)-4-methyl-2H-chromen-2-one
5-(4-tert-butylphenyl)pyrimidine
N,N-dimethyl-2-[methyl({[5-(1H-pyrazol-3-yl)furan-2-yl]methyl})amino]propanamide
N-{[7-(dimethyl-1,3-thiazole-5-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-fluorobenzamide
[(3R,4R)-1-(2-fluoro-4-methylbenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
N-[(2R,3R)-2-ethoxy-1'-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-butyl-2-(furan-2-yl)-N-(furan-2-ylmethyl)-2-oxoacetamide
methyl 3-(4-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
3-[(1R,3R)-3-aminocyclopentyl]-1-[(3-methylphenyl)methyl]urea
6-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1H-indole
2-(2-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
1-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
(2R,3R)-3-amino-1'-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-3,4-dimethoxybenzamide
(3aS,6aS)-2-[(2-fluorophenyl)methanesulfonyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-[4-(trifluoromethyl)benzoyl]pyrrolidin-3-amine
2-chloro-4-[1-methyl-5-(piperidin-1-yl)-1H-1,2,4-triazol-3-yl]benzamide
N-[(4-fluorophenyl)methyl]-4-methyl-5-{1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
5-methoxy-9-(thiophene-2-sulfonyl)-1-oxa-9-azaspiro[5.5]undecane
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
4-[(diethylamino)methyl]-5-ethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}furan-2-carboxamide
1-cyclopentyl-4-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]pyrrolidin-2-one
2-({4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
1-ethyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
methyl (2S)-2-{[5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazol-7-yl]formamido}-3-methylbutanoate
1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N-[(2-{4-[5-(methoxymethyl)thiophene-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]oxolane-2-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]acetamide
(1R,5S,8R)-8-(dimethylamino)-N-[4-fluoro-3-(methylcarbamoyl)phenyl]-3-azabicyclo[3.2.1]octane-3-carboxamide