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N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-(2-methoxyethyl)pyrrolidine-3-carboxamide
N-benzyl-N-methyl-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
1-(2-aminopyridine-4-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-{2-[(2-ethylmorpholin-4-yl)methyl]-4-(4-fluorophenyl)phenoxy}acetic acid
1-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-methyl-3-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]urea
N-(4-{[3-(4-methylphenoxymethyl)piperidin-1-yl]methyl}phenyl)acetamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
5-(1-{4-[(benzyloxy)methyl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3,4-thiadiazol-2-amine
N-methyl-N-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)oxan-4-amine
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
6-[(3,5-dimethoxyphenyl)methoxy]-1-(propan-2-yl)-4-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2-(2-methylpropyl)-6-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
9-methoxy-4-(3-methylpyridine-4-carbonyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{3-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-3-oxopropyl}-3,4-dihydroquinazolin-4-one
N4,N4,5-trimethyl-N2-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrimidine-2,4-diamine
5-{[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
(3R,9R)-11-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4,4,4-trifluorobutan-1-one
5-(dimethylamino)-2-[(1-ethylpyrrolidin-2-yl)methyl]-2,3-dihydropyridazin-3-one
3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]propanamide
1-{2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]pyrimidin-4-yl}piperidin-3-ol
3-hydroxy-1-[(3-methylphenyl)methyl]-3-{[(2-methylpropyl)amino]methyl}piperidin-2-one
1-cyclohexyl-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazole
1-[(1-{6-[(3-methylbutyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]amine
1-(carbamoylmethyl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-3-carboxamide
4-(furan-2-ylmethyl)-2-[(4-methoxyphenyl)methyl]morpholine
3-({[(3,5-dimethoxyphenyl)methyl]amino}methyl)-N,N,7-trimethylquinolin-2-amine
2-[5-(2-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]-N-methylethane-1-sulfonamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
N-methyl-4-oxo-5-(4-phenylazepane-1-carbonyl)-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
3-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
8-cyclopropanecarbonyl-2-[(3,5-dimethylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{5-[4-(piperidin-3-ylmethyl)phenyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-ethyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N-[(1S,2R)-2-aminocyclobutyl]-2-methyl-5-sulfamoylbenzamide
N-butyl-2-[1-(3,4-dimethyl-5-sulfamoylphenyl)-N-methylformamido]acetamide
N-ethyl-2-(morpholin-4-yl)-N-(oxan-4-ylmethyl)-2-(pyridin-3-yl)acetamide
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(naphthalen-2-ylmethyl)piperidin-3-yl]propanoate
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl]propanoate
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(pyridin-4-yl)-1,4-diazepan-6-ol
1-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
1-(3-{[(3-chloropyridin-2-yl)amino]methyl}pyridin-2-yl)piperidin-3-ol
4-(2H-1,3-benzodioxol-5-yloxy)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
3-chloro-2-{3-[1-(prop-2-en-1-yl)-1H-pyrazol-3-yl]phenyl}pyridine
4-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-2-one
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-3-propyl-1H-pyrazole-5-carboxamide
1-[(2-methylpyrimidin-5-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
1-[(3-fluorophenyl)methyl]-4-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane