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1-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-3-yl}-2-phenylethan-1-one
1-[(diethylcarbamoyl)methyl]-N-[(1-ethylpyrrolidin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-2-carboxamide
3-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1-[2-(propylsulfanyl)phenyl]urea
N-(1-benzyl-1H-pyrazol-3-yl)-2-[3-(2-fluorophenyl)-1H-pyrazol-1-yl]acetamide
N-[4-({[2-(1-methylpyrrolidin-2-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
N-[1-(3-chlorophenyl)cyclopropyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-{6-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]pyridin-2-yl}ethan-1-ol
2-(2-hydroxyethyl)-9-[2-(1H-pyrazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-[(adamantan-2-yl)amino]-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]{[3-(trifluoromethyl)phenyl]methyl}amine
N-[(3R,4S)-1-(1H-imidazol-4-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-methoxypropanamide
N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}propanamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(furan-2-ylmethyl)-5-methoxy-N-(prop-2-yn-1-yl)benzamide
1-benzyl-3-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]urea
4-[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepan-2-one
(2S,4S,5R)-4-(2,5-dihydro-1H-pyrrole-1-carbonyl)-5-(2-fluorophenyl)-1-methylpyrrolidine-2-carboxylic acid
5-[1-(2-benzyl-1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]-3-methyl-1,2-oxazole
6-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}pyridin-3-ol
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[(3-methoxyphenyl)methyl]piperidine
2-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}propanamide
1-[(5-propylfuran-2-yl)methyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
2-(5-acetylthiophen-3-yl)-1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
(1R,2S,6R,7S)-4-(5-ethyl-1,2-oxazole-4-carbonyl)-4-azatricyclo[5.2.2.02,6]undecane
1-{[3-(3,4-dimethoxyphenoxy)phenyl]methyl}pyrrolidine
3-(1-benzothiophen-7-yl)-1-(cyclopropylmethyl)-6-[(1R,2S)-2-propylcyclopropanecarbonyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-(4-tert-butylphenyl)-3-(pyrrolidine-1-carbonyl)pyridine
5-(furan-3-carbonyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-{[(1-methyl-1H-imidazol-2-yl)methyl]({[4-(trifluoromethyl)phenyl]methyl})amino}ethan-1-ol
N-[4-fluoro-3-({[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]carbamoyl}amino)phenyl]propanamide
2-(3-methylphenyl)-1-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(morpholin-4-yl)propyl]benzamide
1-butyl-5-(4-methyl-1,3-oxazol-5-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-5-propyl-1,2-oxazole
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(methoxymethyl)piperidine
ethyl 4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)benzamide
1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methoxy-2-methylpropan-1-one
4-(5-acetyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
4-methyl-7-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)-2H-chromen-2-one
(4aS,7aR)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(5-fluoro-2-methylphenyl)methyl]benzamide
(4aS,7aR)-1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
3-{3-[1-(1,4-dioxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-2,5-dimethylpyrazine
2-methoxy-N-(2-methyl-1-{7-[(3-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)acetamide
[(3R,4R)-1-(5-methylthiophene-3-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol