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2-({[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(furan-2-ylmethyl)amino)butan-1-ol
N-(1-benzylpiperidin-3-yl)-5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
5-(1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
2-{1-cyclopentyl-4-[(2,3-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
[(3-methyl-1H-pyrazol-5-yl)methyl][(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amine
9-methoxy-3-[(4-methoxy-3-methylphenyl)methyl]-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(1S,2R)-2-(cyclooctylamino)cyclobutyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-N-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
N,1,4,6-tetramethyl-2-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-dihydropyridine-3-carboxamide
2-{2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
3-{1-[1-(3,5-dimethylphenyl)piperidin-4-yl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-1λ6-thiomorpholine-1,1-dione
2,3,6-trifluoro-N-{[8-(furan-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
N-{2-[(5-methyl-1,3-oxazol-4-yl)formamido]ethyl}pyridine-3-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-methylazepane-2-carboxamide
1-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(pyridin-4-yl)ethan-1-one
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-[2-methoxy-5-({[2-(4-methylphenyl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
6-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]quinoline
2-{[(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
7-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
(3R,4R)-N-butyl-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carboxamide
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-1-[4-(3-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]ethan-1-one
(4aS,7aR)-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
N-(3-methoxypropyl)-6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
9-methoxy-4-[(4-methoxy-2,5-dimethylphenyl)methyl]-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-(3-methyl-1-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
2-(4-{[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}cyclohexyl)-1H-1,3-benzodiazole
N-[(3R,4S)-1-[(3-cyanophenyl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
3-(furan-2-yl)-1-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
4-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetyl}-1-phenylpiperazin-2-one
N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-amine
5-methyl-5-phenyl-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
7-[(3,4-difluorophenyl)methyl]-2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane
(3S,5R)-1-(3-methylbut-2-en-1-yl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
4-(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)-1-[(3-methoxyphenyl)methyl]piperidine
2-[1-(3-fluorophenyl)-5-[(3R)-1,2,3,4-tetrahydroisoquinolin-3-yl]-1H-1,2,4-triazol-3-yl]acetamide
2-(1H-pyrazol-1-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]acetamide
(5S,9aS,9bS)-5-[4-(benzyloxy)phenyl]-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(6-methoxypyridin-3-yl)-N,N,5,6-tetramethylpyrimidin-2-amine
methyl (2R,4S)-1-[2-(1H-1,3-benzodiazol-2-yl)acetyl]-4-hydroxypiperidine-2-carboxylate
(4aS,7aR)-1-[(2-ethoxyphenyl)methyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,3,4,9-tetrahydro-1H-carbazole
7-amino-4-(2,3,4-trimethoxyphenyl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
N-[(4-fluorophenyl)methyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
3-(5-{[3-(2-phenylpyridin-4-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)prop-2-yn-1-ol