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2-[(3R,4S)-3-[(4,6-dimethylpyrimidin-2-yl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-N,N-dimethylacetamide
3-(1H-1,3-benzodiazol-2-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]propanamide
3-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(hydroxymethyl)-1,3-oxazolidin-2-one
N2,N2-dimethyl-6-({[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)-1,3,5-triazine-2,4-diamine
4-(propan-2-yl)-2-{[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]methyl}morpholine
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[(4-methylphenyl)methyl]-1,2-oxazole-3-carboxamide
3-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-1-(2-hydroxyethyl)urea
N-(2-hydroxypropyl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
2,2-dimethylpropyl 2-(1-acetylpiperidin-4-yl)-2,7-diazaspiro[4.5]decane-7-carboxylate
7-{[2-(2-hydroxyethoxy)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
5-(methoxymethyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]thiophene-2-carboxamide
1-[(1-benzyl-1H-imidazol-5-yl)methyl]-4,4-dimethylpyrrolidin-2-one
1-(2-methoxyphenyl)-4-(1-phenylmethanesulfonylpiperidin-3-yl)piperazine
N-(3-methylphenyl)-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-[(cyclohexylmethyl)amino]pyrrolidine-2-carboxamide
1-methyl-3-(2-methylpropyl)-N-[(3R)-pyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
4-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-cyclopropyl-4-methoxy-3-[(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)oxy]benzamide
N-(2-fluorophenyl)-8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
(1R,3S,5S)-8-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-8-azabicyclo[3.2.1]octan-3-ol
1-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)-N-[(4-methylphenyl)methyl]pyrrolidine-1-carboxamide
N-[3-(3-{[cyclohexyl(methyl)amino]methyl}phenoxy)propyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amine
1-{4-[4-({[4-(1H-pyrazol-1-yl)phenyl]methyl}amino)piperidin-1-yl]benzoyl}piperidin-3-ol
1-[2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]imidazolidin-2-one
2-{[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})amino}ethan-1-ol
N-ethyl-7-[(2-phenoxyethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
8-(oxolane-3-carbonyl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
benzyl[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
5-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
5-(4-hydroxy-4-phenylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]piperidin-2-one
ethyl 5-(2-methylpropanoyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(2,3-dihydro-1H-inden-2-yl)-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
9-{[3-(4-methoxyphenoxy)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
N-[2-(N-methylmethanesulfonamido)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-{4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1-(cyclopropylmethyl)piperazin-2-yl}ethan-1-ol
3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
1-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
1-[2-(methylamino)pyridine-4-carbonyl]-3-(2-methylphenyl)pyrrolidin-3-ol
4-(1H-pyrazol-3-yl)-6-(trifluoromethyl)-1H-1,3-benzodiazole
(2S,4R)-4-(3-fluoro-4-methylbenzamido)-1-(3-methylbut-2-en-1-yl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[3-chloro-5-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
6-[3,5-difluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyrazine-2-carboxamide
N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
1-ethyl-3-[4-(piperidin-1-ylmethyl)piperidin-1-yl]piperidine
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-6-aminopyridine-2-carboxamide
7-(furan-3-carbonyl)-N-(2-methoxyethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine