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2-(4-fluorophenoxy)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-{1-[1-(3-chloro-4-ethoxybenzoyl)piperidin-4-yl]ethyl}morpholine
(3aS,6aS)-2-[(2-chloro-4-fluorophenyl)methyl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[cyclohexyl(methyl)amino]-3-(2-{[(3-hydroxypropyl)amino]methyl}phenoxy)propan-2-ol
5-{1-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1H-imidazol-2-yl}-2-methoxyphenol
1-(carbamoylmethyl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
3-[4-methoxy-3-(trifluoromethyl)phenyl]-1H-pyrazole
2-[2-({2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}methyl)phenoxy]acetic acid
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(4-phenylbenzoyl)piperidine
N4-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-N2,N2,6-trimethylpyrimidine-2,4-diamine
2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]acetamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)acetamide
N-[(3R,4S)-4-cyclopropyl-1-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]pyrrolidin-3-yl]acetamide
4-{[2-(dimethylamino)ethyl]({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)carbamoyl}pyridin-1-ium-1-olate
(2S)-5-oxo-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]pyrrolidine-2-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
1'-[(3-hydroxyphenyl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
5-(naphthalen-2-yl)-3-[4-(2-phenoxyethyl)piperazin-1-yl]-1,2,4-triazine
N-[3-(1,3-benzoxazol-2-yl)propyl]-2,3-dimethylquinoxaline-6-carboxamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl}propanamide
8-cyclobutyl-3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(2-methoxyethyl)piperidine-3-carboxylate
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-[4-(2-phenylethyl)morpholin-3-yl]acetamide
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
methyl 4-{4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}benzoate
N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-6-(morpholin-4-ylmethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
{1-[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}methanol
5-[1-(3,4-difluorobenzoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
1-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(1-methyl-3-phenyl-1H-pyrazol-5-yl)urea
methyl 4-[6-amino-5-cyano-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)pyridin-2-yl]-5-methylfuran-2-carboxylate
9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
4-{[({4-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)amino]methyl}hepta-1,6-dien-4-ol
1-(3-chloro-4-methoxyphenyl)-N-(1H-imidazol-2-ylmethyl)-N-methyl-5-oxopyrrolidine-3-carboxamide
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[3-(pyridin-3-yl)propyl]propanamide
3-cyclopropyl-5-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-phenyl-1H-1,2,4-triazole
6-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
2-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-4-hydroxyquinoline-6-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-(quinoline-8-carbonyl)pyrrolidine-3-carboxylic acid
N-(2-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methylbenzamide
8-(1,5-dimethyl-1H-indazole-3-carbonyl)-1-oxa-8-azaspiro[4.5]decane
N-({2-[4-(morpholin-4-yl)butoxy]phenyl}methyl)pyrrolidin-3-amine
1-(5-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methylphenyl)imidazolidin-2-one
N-{[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
6-(benzyloxy)-4-(4-phenylbutanoyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
4-{3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
methyl 4-(methylsulfanyl)-2-({4-[4-(pyridine-3-amido)-1H-pyrazol-1-yl]phenyl}formamido)butanoate
ethyl 1-(3-phenylprop-2-ynoyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
5-methyl-2-(thiophen-2-yl)-4-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1,3-oxazole