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1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-4-phenylbutane-1,2-dione
1-(4-methylquinazolin-2-yl)-N-(1-phenylcyclopropyl)pyrrolidine-2-carboxamide
4-{4-[2-(3-fluorophenyl)acetyl]piperazin-1-yl}-2-methyl-2,3-dihydro-1H-isoindole-1,3-dione
1-cyclopropyl-3-(4-methoxyphenyl)-3-(2-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)pyrrolidine-2,5-dione
(4aS,8aR)-1-(3-aminopropyl)-6-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-[(4-chlorophenyl)methyl]-N-[2-(6-methylpyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(2-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)ethan-1-ol
N-[(2R,3R)-2-methoxy-1'-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
(3S,4S)-4-(3-methoxyphenyl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-3-ol
4-(4-cyclopropanecarbonyl-6-hydroxy-1,4-diazepan-1-yl)-2-methoxypyridine-3-carbonitrile
5-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(3S)-N,N-dimethyl-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]azepan-3-amine
4-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-N-(1-methyl-1H-pyrazol-4-yl)benzamide
2-methyl-4-{5-[1-(1,2-oxazol-5-ylmethyl)-4-phenyl-1H-imidazol-5-yl]thiophen-2-yl}but-3-yn-2-ol
1-cyclopentyl-4-(4-methylpyrimidin-2-yl)piperazin-2-one
3-{[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(6-{pyrazolo[1,5-a]pyridin-7-yl}pyridin-3-yl)methyl]morpholine
2-(4-acetylpiperazin-1-yl)-2-[4-(methylsulfanyl)phenyl]acetic acid
1-[5-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazine-1-carbonyl)thiophen-2-yl]ethan-1-one
6-methoxy-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrimidin-4-amine
2-(6-aminopyridin-3-yl)-2-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}acetic acid
8-(furan-2-ylmethyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(oxan-4-yl)thieno[2,3-d]pyrimidin-4-amine
N-[(1R,2R)-2-hydroxycyclohexyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-propylacetamide
N,N-dimethyl-5-[4-(piperidin-1-yl)butanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(6-fluoro-4-methylquinazolin-2-yl)-N-[(1-hydroxycyclohexyl)methyl]pyrrolidine-2-carboxamide
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-3-chlorobenzamide
N-[(3R,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-5-methylpyrazine-2-carboxamide
5-methyl-4-[(4-methyl-1H-imidazol-1-yl)methyl]-2-[4-(methylsulfanyl)phenyl]-1,3-oxazole
9-cyclopentanecarbonyl-2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-(3-{[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
(1S,5R)-6-(5-chloronaphthalene-1-carbonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
7-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-cyclopropyl-N-({4-[3-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)propoxy]phenyl}methyl)thiophene-2-carboxamide
N,N,4-trimethyl-5-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}pyrimidin-2-amine
(2S,4R)-1-benzyl-N-ethyl-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetamido]pyrrolidine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}piperidin-1-yl)benzamide
4-chloro-1-ethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
N'-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N'-[2-(cyclohex-1-en-1-yl)ethyl]-N,N-dimethylbutanediamide
N-[(4-chlorophenyl)methyl]-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
1-(4-methylpiperazin-1-yl)-3-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]propan-1-one
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
5-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-[(2R,3R)-2-hydroxy-1'-[(3-hydroxy-4-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
3-methyl-7-{2-[(2-methylphenyl)sulfanyl]acetyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(4-fluoro-3-methylphenyl)-1-methyl-6-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
methyl (2S)-1-{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}pyrrolidine-2-carboxylate
1-(2-cyclohexylethyl)-3-hydroxy-3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)piperidin-2-one
3-({1-[3-(3-fluorophenyl)propanoyl]pyrrolidin-3-yl}methyl)benzamide
3-[5-({[(2-methylphenyl)methyl](2-methylpropyl)amino}methyl)thiophen-3-yl]prop-2-yn-1-ol