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3-propyl-N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}morpholine-4-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]acetamide
2-{1-cyclopentyl-4-[(3-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-(1-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)pyridin-2-amine
N-[1-(4-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]pyridine-3-carboxamide
1-[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-4-oxo-3,4-dihydroquinazoline-2-carboxamide
3-(3-methoxyphenyl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-ethyl-1-[9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
6-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
N-(3-cyanophenyl)-2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-(1-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-imidazol-2-yl)phenol
1-tert-butyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-5-oxopyrrolidine-3-carboxamide
[2-(pyridin-3-yl)ethyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
(4aS,8aR)-6-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
1-[1-(3-phenylpropyl)piperidin-4-yl]-N-[(2S)-pyrrolidin-2-ylmethyl]piperidine-4-carboxamide
N-[(2,4-difluorophenyl)methyl]-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
4-[4-(4-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}piperidin-1-yl)benzoyl]morpholine
ethyl 2-(4-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}phenyl)acetate
1-{2-[2-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
1-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
(3R,4R)-N-[(2-fluorophenyl)methyl]-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carboxamide
N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopentanecarboxamide
1-ethyl-N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine-2-carboxamide
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(4-fluoro-3-methylphenyl)ethan-1-one
2-ethyl-1-methyl-4-(thian-4-yl)piperazine
1-[2-(4-methoxyphenyl)ethyl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
2-oxo-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-1-phenylpyrrolidine-3-carboxamide
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyridin-2-amine
(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-1H-1,2,4-triazole-5-carboxamide
N,1,3-trimethyl-N-[2-(morpholin-4-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-amino-4-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]quinolin-8-ol
2-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-[(pyridin-2-ylmethyl)amino]benzamide
1-[3-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl)phenyl]pyrrolidin-2-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-2-(2,5-dioxoimidazolidin-1-yl)-N-methylacetamide
methyl (2S)-1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}pyrrolidine-2-carboxylate
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]cyclopropane-1-carboxamide
1-[3-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
1-{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine
4-(benzyloxy)-1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{2-[6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidin-4-yl]ethyl}acetamide
4-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}morpholine-2-carboxylic acid
N-(1,3-benzothiazol-2-ylmethyl)-2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)benzamide