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3-propyl-1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]piperidine-3-carboxylic acid
2-({[(2-chloro-6-fluorophenyl)methyl](ethyl)amino}methyl)pyridine-3-carboxylic acid
7-(1,3-benzothiazol-2-yl)-4-[3-(dimethylamino)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-1-[(2-fluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-(pyrimidin-5-ylmethyl)pyrrolidin-3-amine
4-[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]morpholine
N-[4-(4-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}piperidin-1-yl)phenyl]-5-phenylpentanamide
5-phenyl-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2-oxazole-3-carboxamide
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(piperidin-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]propanamide
4-chloro-5-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}-N,N-dimethyl-1,3-thiazol-2-amine
1-(azepan-1-yl)-3-[3-({[3-(1H-indazol-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
2-(pyridin-4-ylmethyl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
2-amino-6-(1-methyl-1H-pyrrol-3-yl)-4-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
N-{2-[1-(5-fluoro-2-methoxyphenyl)-1H-imidazol-4-yl]ethyl}acetamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-N-(propan-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]propanamide
2-(diethylamino)-N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}acetamide
N-cyclopentyl-N'-[2-(pyridin-3-ylformamido)ethyl]butanediamide
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(oxan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(2R,3R)-1'-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
N-[2-(azepan-1-yl)-2-phenylethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-[(3R,4R)-1-(5-chlorothiophene-2-carbonyl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
N-(1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
ethyl 4-benzyl-1-[(2,3-dimethoxyphenyl)methyl]piperidine-4-carboxylate
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-[2-(1H-imidazol-4-yl)ethyl]-4-methyl-7-(methylsulfanyl)quinolin-2-amine
5-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]-1,3-dimethylimidazolidine-2,4-dione
(3aR,6aR)-N-[2-(azepan-1-yl)ethyl]-2-cyclopropanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylacetamide
2-(3,4-dimethoxyphenyl)-1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-({7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzenesulfonamide
2-(benzyloxy)-1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]ethan-1-one
N-(1-methyl-1H-1,2,3-triazol-4-yl)-2-(4-methyl-1H-indol-1-yl)acetamide
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-imidazol-1-yl)butan-1-one
4-[(2S,3R)-2-amino-3-hydroxybutanoyl]-1-(2-chlorophenyl)piperazin-2-one
2-(dimethylamino)-N-[3-methyl-1-(7-{2-[3-(trifluoromethyl)phenyl]acetyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)butyl]acetamide
11-[(cyclopropylmethyl)amino]-4-[(2-methoxynaphthalen-1-yl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(2-hydroxyphenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrazole-5-carboxamide
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-1,2,4-triazole-5-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
N-{[2-(2-cyclobutaneamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-oxopyrrolidin-1-yl)benzamide
3-{[4-(3-chlorophenyl)-5-({[(3,4-difluorophenyl)methyl](methyl)amino}methyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
1-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
methyl 7-oxo-3-[3-(piperidin-1-yl)propanoyl]-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(2-methylpyridin-4-yl)-4-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]-1,4-diazepane
5-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
7-(3-chlorophenyl)-9-[(1-methylpiperidin-3-yl)methoxy]-4-(thiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S)-4-methyl-2-{[2-(trifluoromethyl)pyrimidin-4-yl]amino}pentanamide