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1-(pyrrolidin-1-yl)-2-(4-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-one
1'-(5-methoxy-1H-indole-2-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-[(3-hydroxyphenyl)methyl]-N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[1-(3-methylbutyl)-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl]ethan-1-ol
1-(benzyloxy)-8-(4-phenylbenzoyl)-1,8-diazaspiro[4.5]decan-2-one
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}-N-[1-(thiophen-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-(1-hydroxybutan-2-yl)-N-(thiophen-3-ylmethyl)cyclopropanecarboxamide
2-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}acetic acid
2-methyl-N-(1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-[4-(furan-2-yl)phenyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidine-3-carboxamide
N-[(2,5-difluorophenyl)methyl]-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
3-[2-(dimethylamino)ethyl]-5-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
N-{[1-(quinolin-2-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}furan-2-carboxamide
2-(4-{[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
N-benzyl-3-[1-(dimethylsulfamoyl)piperidin-4-yl]-N-methylpropanamide
1-(2-oxo-2-{spiro[azepane-4,2'-chromene]-1-yl}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
[3-(3-phenylpropyl)piperidin-3-yl]methanol
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
(3S,5R)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
3-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-ethylpropanamide
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-methylpropanamide
1-(2-methoxyacetyl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
(4aR,8aS)-1-[3-(dimethylamino)propyl]-6-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-decahydro-1,6-naphthyridin-2-one
6-(cyclopropylmethoxy)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-[1-(pyridin-2-yl)piperidine-3-carbonyl]-1,4-diazepan-2-one
3-{1-[(1,2-dimethyl-1H-indol-3-yl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
(1S,4S)-5-(ethanesulfonyl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-[2-(dimethylamino)ethyl]-5-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
1-(4-benzylpiperazin-1-yl)-3-[1-(1H-indol-3-ylmethyl)piperidin-3-yl]propan-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-6-azaspiro[2.5]octane-1-carboxamide
5-(4-acetylphenoxymethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-[4-(2-hydroxypropan-2-yl)piperidin-1-yl]-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
2-methoxy-N-({8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
1-({3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)azocane
4-[(2-aminopyridin-3-yl)methyl]-1-methylpiperazine-2-carboxylic acid
1-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}phenyl)-1H-pyrazole
methyl 4-[(3-{2-[(1-methylpiperidin-3-yl)formamido]ethyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)methyl]benzoate
2-[2-(ethylamino)pyrimidin-5-yl]-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
3-benzyl-8-[(2-hydroxy-3-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-6-(cyclobutylmethyl)-3-{[3-(morpholin-4-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2-[1-(cyclohex-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}-3-fluoro-4-methylbenzamide
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-[3-(2-methylphenyl)-1H-pyrazol-1-yl]acetamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
3-({[(2-chloro-4-fluorophenyl)methyl]amino}methyl)-N,N-dimethylpyridin-2-amine
(3R,4S)-4-cyclopropyl-1-(5-fluoro-1-methyl-1H-indole-2-carbonyl)pyrrolidin-3-amine
3-(1-methyl-1H-1,3-benzodiazol-5-yl)-1-[2-(4-phenylpiperidin-1-yl)ethyl]urea
3-(3-methylphenyl)-1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
2-{1-[(2-ethoxyphenyl)methyl]-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide