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2-{[(6-methoxypyridin-3-yl)methyl](thiophen-3-ylmethyl)amino}butan-1-ol
2-(2-methoxyethyl)-9-(5-methylthiophene-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]{[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]methyl}amine
(1S,5R)-N-(3-cyanophenyl)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-(piperidine-1-carbonyl)-1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidine
1-cyclopropanecarbonyl-2-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]piperidine
3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]-5-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
2-{1-[(4-methylphenyl)methyl]-4-propylpiperazin-2-yl}ethan-1-ol
1-[2-(benzyloxy)benzoyl]-3-(1H-imidazol-2-yl)piperidine
N-butyl-3-[2-(methylsulfanyl)benzoyl]piperidine-1-carboxamide
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-sulfamoylbenzamide
8-[2-(4-chlorophenyl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,3-thiazol-2-ylmethyl)acetamide
6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]pyrrolidin-3-yl]acetamide
6-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[4-methyl-6-({2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}amino)pyrimidin-2-yl]phenol
N-methyl-5-({[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}methyl)furan-2-carboxamide
5-(1H-indol-4-yl)-1,2,3,4-tetrahydroisoquinoline
3-{methyl[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}-1-phenylpropan-1-ol
N-phenyl-3-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}benzamide
(4aS,8aR)-6-(3-fluoropyridin-2-yl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
8-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[4-(difluoromethoxy)benzoyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(2-ethyl-5-oxopyrrolidin-2-yl)-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]propanamide
N-[(2R,3R)-1'-(2,3-difluorobenzoyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
(2S,4S)-4-amino-1-[6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-benzyl-9-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-6-[2-(methylamino)pyrimidine-5-carbonyl]-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(3-phenylpropyl)piperidin-4-yl)methanol
N6-cyclopentyl-N5-methyl-N5-[1-(1,3-thiazol-2-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
methyl 1-{2-hydroxy-3-[3-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
1-cyclopentyl-4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
2-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzonitrile
3-cyclopentyl-5-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
4-methyl-2-{[4-(4-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenol
N-cyclopropyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-3-(thiophen-3-yl)propan-1-one
3-({1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
2-(3,5-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
1-({4-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)azetidin-3-ol
4-[(3R,4S)-3-[(2-methylpyrimidin-4-yl)amino]-4-(propan-2-yl)pyrrolidine-1-carbonyl]oxane-4-carbonitrile
3-[(4-fluorophenyl)methyl]-N-[2-(methylsulfanyl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
methyl 1-ethoxy-8-(2-ethylbutyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-6-methoxy-1-methyl-1H-indole
N-[1-(3-methylpyridin-2-yl)ethyl]-4-oxo-3,4-dihydroquinazoline-2-carboxamide
(1S,6R)-9-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
6-benzoyl-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
N-[(3R,4R)-3-hydroxy-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl]pyridine-3-carboxamide