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N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
2-[1-(2-methylpropyl)-4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
5-benzyl-N-[1-(furan-2-yl)ethyl]-N-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,4-dimethyl-2-(propan-2-yl)pyrimidine-5-carboxamide
1-ethyl-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperazin-2-one
N-(2H-1,3-benzodioxol-5-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-amine
N-(oxolan-2-ylmethyl)-3-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}propanamide
1-[cyclohexyl(thiophen-2-yl)methyl]-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
(3R)-1-[3-(4-methylphenyl)benzoyl]pyrrolidin-3-ol
5-[(isoquinolin-5-yloxy)methyl]-N-[2-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
6-[3-(4-fluorophenoxymethyl)piperidin-1-yl]pyridine-2-carboxylic acid
N-[3-(1H-indol-1-yl)propyl]-3-propanamidobenzamide
3-cyclopropyl-5-(2-phenyl-1H-imidazol-4-yl)-1H-1,2,4-triazole
2-[({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)amino]pyridine-4-carboxamide
methyl[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl](oxolan-3-ylmethyl)amine
N-[(1-hydroxycyclohexyl)methyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
6-tert-butyl-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
[(3R,4R)-1-(1,3-benzothiazol-2-yl)-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
5-chloro-N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
9-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-({[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]amino}methyl)benzoate
N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[2-(methylsulfanyl)ethyl]propanamide
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-fluorophenyl)urea
1-cyclopentyl-5-oxo-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-3-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
4-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-2-methylphenol
1-cyclopropanecarbonyl-N-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-4-carboxamide
N-{1-[7-(furan-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-methoxypropanamide
5-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-ethyl-1'-(quinolin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(4-chloro-1H-pyrazol-1-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
ethyl 1-(3-phenylpropyl)-5-[2-(pyrimidin-2-ylsulfanyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-ethyl-3-{1-[3-(1H-pyrazol-5-yl)phenyl]-1H-imidazol-2-yl}piperidine
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-(1-methoxypropan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}dimethylamine
2-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}phenol
N-[(3S,4R)-1-[2-(4-acetylphenoxy)acetyl]-4-propylpyrrolidin-3-yl]acetamide
N-ethyl-7-fluoro-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(2-methylpyrimidin-5-yl)quinoline-4-carboxamide
2-[(5-chloro-2-fluorophenyl)methyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-[2-(3-chlorophenoxy)ethyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]imidazo[1,2-a]pyrimidine-2-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-methyl-1,3-oxazole-4-carboxamide
2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-3-ol
N-{[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-3-yl]methyl}butanamide
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(4-{thieno[2,3-d]pyrimidin-4-yl}-1H-pyrazol-1-yl)acetamide
5-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione