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2,4-dioxo-N-[1-(pyridin-4-yl)propan-2-yl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-(furan-2-ylmethyl)-5-(1-propanoylpiperidin-4-yl)-5-propylimidazolidine-2,4-dione
1-[3-(methoxymethyl)pyrrolidin-1-yl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butan-1-one
4-(4-methoxyphenyl)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-oxobutanamide
N-ethyl-5-methyl-4-{[2-(morpholin-4-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-(4-pentanamidophenyl)-4-(propan-2-yl)-1,2,3-thiadiazole-5-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
7-{2-[(4-chlorophenyl)sulfanyl]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-(thiophen-2-ylmethyl)acetamide
3-({8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decan-1-yl}methyl)phenol
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-(pyridin-4-yl)propanamide
7-methanesulfonyl-4-methyl-2-[4-(morpholin-4-yl)piperidin-1-yl]quinazoline
1,3-dimethyl-N-(2-propoxyethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(2,5-dimethoxyphenyl)-N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]acetamide
1-[3-(2-methylphenoxy)azetidin-1-yl]-2-(pyridin-2-ylsulfanyl)propan-1-one
5-[(3-methoxyphenyl)methyl]-3-methyl-5-{1-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[2-(2,3-dimethoxyphenyl)ethyl]-3-azaspiro[5.5]undecan-9-amine
1-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(1H-indazol-7-yl)urea
ethyl 3-(2-methoxyethyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxylate
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}morpholine
2-(2-{1-[3-(thiophen-2-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
2-[(4-methoxyphenyl)methyl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
2-amino-4-(3-hydroxyphenyl)-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
N-(furan-2-ylmethyl)-3-[methyl(quinolin-3-ylmethyl)amino]propanamide
1-(2,3-dihydro-1H-inden-2-yl)-N-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-amine
2-ethyl-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N3-cyclooctyl-N5-[(3-fluoro-4-methylphenyl)methyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
(5S,9aS,9bS)-5-(1-benzofuran-2-yl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[7-(3-chloro-2-fluorobenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}oxolane-3-carboxamide
4-(1-{4-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-1H-1,2,3-triazol-1-yl}ethyl)pyrimidine
ethyl 1-(dimethylsulfamoyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
5-methyl-3-(3-oxo-3-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}propyl)-2,3-dihydro-1,3-benzoxazol-2-one
3,5-difluoro-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}pyridine-2-carboxamide
(2S,4S)-1-benzyl-4-{[(5-chloro-2-hydroxyphenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
2-(but-2-yn-1-yl)-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-chloro-1H-pyrazole-3-carboxamide
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-[(6-fluoroquinolin-2-yl)methyl]pyrrolidin-3-yl]methanol
5-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
5-(2,5-dimethylfuran-3-yl)-3-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-1,2,4-triazine
3-{5-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
4-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-indole
2-(2-methylpropyl)-8-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(2-methoxynaphthalen-1-yl)ethyl]-2-(methylamino)acetamide
3-hydroxy-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)pyridine-2-carboxamide
5-acetamido-1-(2-methoxyethyl)-2-(pyridin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-1,3-benzodiazole-7-carboxamide
methyl 3-({[1-(4-chlorophenyl)cyclobutyl]formamido}methyl)-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate