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5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]pyridin-2-amine
(5S)-5-{[(pyridin-4-ylmethyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amino]methyl}pyrrolidin-2-one
2-(ethylamino)-N-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]pyrimidine-5-carboxamide
3-(2H-1,3-benzodioxol-4-ylmethyl)-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)(naphthalen-2-ylmethyl)amine
N-[2-methyl-1-(pyridin-2-yl)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(1-{1-[1-(2-fluorophenyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
2-[2-benzyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]-N-methylacetamide
N-(3-{[butyl(furan-2-ylmethyl)carbamoyl]amino}-4-fluorophenyl)propanamide
5-[(2,2-dimethyloxan-4-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
7-(cyclopropylmethyl)-N-[(2-methylphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
N'-(cyclohex-1-en-1-ylmethyl)-N-[2-(methylsulfanyl)phenyl]butanediamide
N-[(3R,4S)-1-(2-methoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)-1,3-thiazole-5-carboxamide
1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
2-(naphthalen-2-yloxy)-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]propan-1-one
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(morpholin-4-yl)ethyl]acetamide
9-methoxy-7-(5-methylthiophen-2-yl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{4-[1-(dimethylamino)ethyl]phenyl}-N,6-dimethylpyrimidin-4-amine
N-{2-[2-(2,5-dioxoimidazolidin-1-yl)acetamido]-4-methylphenyl}pentanamide
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4-(2,6-dimethylpyridin-4-yl)piperazine
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluorobenzamide
3-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propanoic acid
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
N2-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-fluoro-N4-methylpyrimidine-2,4-diamine
3-(4-methylphenyl)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
[3-(1H-imidazol-1-yl)propyl]({[6-methyl-2-(prop-2-en-1-yloxy)quinolin-3-yl]methyl})amine
1-[2-(dimethylamino)ethyl]-N-(diphenylmethyl)-6-oxopiperidine-3-carboxamide
N-[(3R,4S)-1-(2-methyl-5-propylpyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(methylamino)acetamide
2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-N-[(2-methoxyphenyl)methyl]acetamide
2-cyclopentyl-9-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-cyclopentanecarbonyl-N-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]piperidine-4-carboxamide
1-cyclohexyl-4-[4-(methylsulfanyl)benzoyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-(cyclopropylmethyl)-1-ethyl-N-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(2-fluorophenyl)methyl]-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(4-chlorophenyl)methyl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[3-(pyridin-4-yl)propyl]acetamide
1-cyclopentyl-3-(2-fluorophenyl)-3-[2-oxo-2-(3-propanoylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione
1-{[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}azocane
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-(1,4-oxazepan-4-yl)butan-1-one
2-{4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]morpholin-3-yl}acetic acid
2,5,6-trimethyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidin-4-amine
1-{4-[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amino]piperidin-1-yl}ethan-1-one
2-(pyrrolidin-3-yl)-N-(quinolin-3-yl)benzamide
N-(cyclopropylmethyl)-1-(4,7-dimethylquinazolin-2-yl)-N-(oxolan-2-ylmethyl)piperidine-3-carboxamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1,4-diazepane
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-propylacetamide
(1R,5R)-6-[2-methyl-2-(morpholin-4-yl)propyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
8-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one