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(2R,3S,6R)-5-(2H-1,3-benzodioxole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]-8-azabicyclo[3.2.1]octane
(2E)-3-phenyl-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-(3-hydroxyphenyl)-N-methyl-5-oxopyrrolidine-3-carboxamide
6-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)pyridine-2-carboxylic acid
3-methyl-7-[1-(2-phenylethyl)piperidin-4-yl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methyl-1H-1,3-benzodiazole-6-carboxamide
1,5,6-trimethyl-3-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1,2-dihydropyridin-2-one
1-({4-[(3-chlorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-4-ol
4-(2-methylphenoxy)-1-(pyrazin-2-yl)piperidine-4-carboxylic acid
methyl 4-{7-[(2,3-difluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-4-oxobutanoate
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2,2-dimethylpropan-1-one
N-benzyl-N-(cyclobutylmethyl)-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-(methoxymethyl)-N-[4-(5-methyl-4-{[3-(5-methyl-1H-pyrazol-1-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]furan-2-carboxamide
2-[5-cyclopropyl-4-(4-methylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(2,5-dimethoxyphenyl)pyrimidine
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methylbenzamide
3-[4-(3-chlorophenyl)piperazine-1-carbonyl]-1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
N-(1-{4-[4-(quinazolin-4-yl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)furan-3-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-[(1-methylpiperidin-3-yl)methyl]-2-phenoxy-N-(2-phenylethyl)acetamide
N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
(1R,5R)-3-benzoyl-6-(1H-imidazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-2-phenylpyrimidine
3-{[4-(2-chlorophenyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-(quinolin-8-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-(4-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)-1λ6-thiolane-1,1-dione
1-[1-methyl-5-({methyl[3-(oxolan-2-yl)propyl]amino}methyl)-1H-pyrrol-3-yl]ethan-1-one
N-[1-(pyrimidin-4-yl)ethyl]-4-(trifluoromethyl)pyrimidin-2-amine
1-cyclopentyl-4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]piperazine
5-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-2-(3-methylphenyl)pyrimidin-4-ol
2-(2-oxopyrrolidin-1-yl)-N-[(3R,4S)-4-(propan-2-yl)-1-(pyridin-4-yl)pyrrolidin-3-yl]acetamide
N-(oxan-4-ylmethyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
3-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-9-methoxy-N-(3-methylbutyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-ethyl-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(pyridin-4-ylmethyl)propanamide
2-[({1-[5-(phenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
(2S,4R)-4-amino-N-[2-(2-ethoxyphenyl)ethyl]pyrrolidine-2-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}phenyl)-3H,4H,5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-one
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide
3-(3-fluorophenyl)-3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
2-{2-[4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2,3,4-tetrahydrophthalazine-1,4-dione
ethyl 3-[(3-methoxyphenyl)methyl]-1-[3-(1H-pyrazol-4-yl)propanoyl]piperidine-3-carboxylate
6-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-2-carboxylic acid
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
(2E)-4-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}pent-2-enamide
4-{4-[(4-ethoxyphenyl)methyl]piperazine-1-carbonyl}-1-(propan-2-yl)pyrrolidin-2-one
3-(1,2-oxazinan-2-yl)-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]propan-1-one
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
2-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}quinolin-8-ol