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(3R,5R)-N-butyl-1-(2-phenylethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)methylamine
4-hydroxy-3-methoxy-N-[(1S,2R)-2-[(1-propylpiperidin-4-yl)amino]cyclobutyl]benzamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-methylfuran-3-carboxamide
ethyl 5-({2-oxo-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-1-yl}methyl)furan-2-carboxylate
4-(azepan-1-yl)-5-methyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N-(1H-imidazol-2-ylmethyl)-6-(4-methoxyphenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(2S)-N-(2,3-difluorophenyl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(1S,5R)-1,3,3-trimethyl-6-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-6-azabicyclo[3.2.1]octane
1-(2-amino-4-phenylpyrimidine-5-carbonyl)-4-(hydroxymethyl)piperidin-4-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-3-yl}propanamide
1-[(3-fluorophenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperazine
N-methyl-1-(2-phenylethyl)-N-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-amine
4-phenyl-3-[(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1-{2-oxo-2-[2-(pyridin-2-yl)piperidin-1-yl]ethyl}-1H-pyrazol-4-yl)benzamide
(1R,5S)-6-methyl-3-{[2-(trifluoromethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2,4-dimethyl-N-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}pyrimidine-5-carboxamide
2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-cyclopropylacetamide
N-cyclopropyl-1-{1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-4-yl}piperidine-3-carboxamide
N,3,5,7-tetramethyl-N-[1-(pyrimidin-4-yl)ethyl]-1H-indole-2-carboxamide
methyl (2S)-2-(3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamido)-4-methylpentanoate
4-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-2,6-dimethylpyrimidine
1-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-{imidazo[1,2-a]pyridin-3-ylmethyl}-3-methyl-1-(1,3,4-thiadiazol-2-yl)urea
6-(cyclopropylmethoxy)-4-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
4-(5-methylpyridin-2-yl)-1-{[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl}piperidin-4-ol
1-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
3-({[(6-hydroxypyrimidin-4-yl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
methyl 2-[8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-[3-(1H-pyrazol-4-yl)propyl]-4-(pyridin-2-ylmethyl)piperazine
ethyl 4-{6-[1-(4-chlorophenyl)cyclopropanecarbonyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(2-methylphenyl)propanamide
2-(5-chloro-2-methoxyphenyl)pyridine-4-carbonitrile
4-hydroxy-1-[3-(4-methoxyphenyl)propanoyl]piperidine-4-carboxylic acid
(2S)-N-[2-(pyridin-3-yloxy)phenyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidine-2-carboxamide
(5Z)-5-[2-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)-2-oxoethylidene]-1,3-thiazolidine-2,4-dione
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-N-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
7-(2-hydroxyethyl)-2-(5-phenyl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-(5-propyl-4H-1,2,4-triazol-3-yl)urea
4-[3-(3,4-difluorophenyl)-1-(6-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]butanamide
2,6-difluoro-N-[(7-{[5-(methoxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}propan-1-one
methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})[2-(oxan-2-yl)ethyl]amine
2-(dimethylamino)-N-{3-methyl-1-[7-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}acetamide
2-{4-[(2-ethylpyrimidin-5-yl)methyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methylpyridin-2-amine
4-{[(1-ethyl-1H-imidazol-5-yl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid