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1-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-4-(4H-1,2,4-triazol-3-yl)piperidine
(2E)-N-cyclopropyl-3-(3-fluorophenyl)-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}prop-2-enamide
5-{[(furan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}-N,N-dimethylpyrimidin-2-amine
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methoxypyridine-3-carboxamide
N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]-N-[3-(oxolan-2-yl)propyl]benzamide
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
4-[3-(3-hydroxy-3-methylbutyl)benzoyl]morpholine-2-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-ethyl-2H-1,3-benzodioxole-5-carboxamide
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-(dimethyl-1,2-oxazole-4-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
ethyl 3-[(1-cyclohexanecarbonylpyrrolidin-2-yl)formamido]propanoate
2-ethyl-9-[4-(4-methylphenyl)-4-oxobutyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 5-(1-methanesulfonylpiperidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
ethyl 5-{[4-(diethylamino)phenyl]methyl}-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1S,3R)-3-amino-N-[(5-chloro-1-benzothiophen-3-yl)methyl]cyclopentane-1-carboxamide
3-benzyl-1-(3-methoxypropyl)-8-(thiophen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{1-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]piperidin-3-yl}benzoic acid
1-[2-(dimethylamino)ethyl]-N-(1-methoxypropan-2-yl)-6-methyl-4-oxo-2-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
N-{[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
N-[(1-cyclohexylpiperidin-3-yl)methyl]-5-(methoxymethyl)-N-(pyridin-3-ylmethyl)furan-2-carboxamide
3-[1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)azetidin-3-yl]pyridine
N-({7-[(2-chloro-6-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
(4aS,7aR)-1-cyclopropanecarbonyl-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-[5-(2-ethoxyethyl)-1,3,4-thiadiazol-2-yl]-3-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]urea
N-(1-{7-[(3,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxybenzamide
2-butyl-8-{7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
4-(1-{[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]amino}ethyl)hepta-1,6-dien-4-ol
1-cyclohexyl-4-(2-methyl-1,3-thiazole-4-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
5-{1-[2-(3-chlorophenyl)acetyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
3-acetamido-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}propanamide
N-{1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-1-oxopentan-2-yl}acetamide
N-(2-ethoxyethyl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}phenol
4-(3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}imidazo[1,2-a]pyridine-2-carbonyl)morpholine
(3R,4R)-3-cyclopropyl-1-(2,3-dihydro-1H-indene-5-carbonyl)-4-methylpyrrolidin-3-ol
4-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-phenylpyrimidine
N-[2-(ethanesulfonyl)ethyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
{2-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-1,3-thiazol-4-yl}methanol
1-[3-({[(2-chlorophenyl)methyl]amino}methyl)-5,6,7-trimethoxyquinolin-2-yl]piperidin-3-ol
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-[(2E)-2-methylbut-2-en-1-yl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(2-chlorophenyl)-1-(3-methoxypropyl)-3-(2-oxo-2-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}ethyl)pyrrolidine-2,5-dione
1-(2-fluorophenyl)-4-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}piperazine
3-ethyl-1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-3-ol
1,5-dimethyl-2-phenyl-4-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}-2,3-dihydro-1H-pyrazol-3-one
1-(morpholin-4-yl)-3-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)propan-1-one
6-chloro-N,N-dimethyl-3-{[4-(3-methylphenoxy)piperidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
4-(4-{[ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenyl)but-3-yn-1-ol